| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| F2 |
2-[3-(5-carbamimidoyl-1H-1,3-benzodiazol-2-yl)-4-hydroxy-5-(3-nitrophenyl)phenyl]acetic acid |
150000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
2-[3-(1H-1,3-benzodiazol-2-yl)-4-hydroxy-5-(3-nitrophenyl)phenyl]acetic acid |
150000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
2-(3-{5-amino-1H-imidazo[4,5-b]pyridin-2-yl}-4-hydroxy-5-(3-nitrophenyl)phenyl)acetic acid |
150000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
6-Chloro-2-(3-cyclopentyloxy-2-hydroxy-phenyl)-1H-benzoimidazole-5-carboxamidine |
165000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
2-(3,4-Dihydroxyphenyl)-5-[[4-[[2-(3,4-dihydroxyphenyl)-3,7-dihydroxy-4-oxochromen-5-yl]oxymethyl]phenyl]methoxy]-3,7-dihydroxychromen-4-one |
NA |
267000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
acetic acid;(2S)-N-[(4-carbamimidoylphenyl)methyl]-1-ethylpyrrolidine-2-carboxamide |
250000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
acetic acid;(2S)-N-[(4-carbamimidoylphenyl)methyl]-1-sulfamoylpyrrolidine-2-carboxamide |
163000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
Octasodium;[2-(3,4-disulfonatooxyphenyl)-5-[[4-[[2-(3,4-disulfonatooxyphenyl)-4-oxo-3,7-disulfonatooxychromen-5-yl]oxymethyl]phenyl]methoxy]-4-oxo-3-sulfonatooxychromen-7-yl] sulfate |
NA |
156000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
Dihydrospumigin M |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
Disodium;[3-ethoxycarbonyl-5-[(3-ethoxycarbonyl-6-methoxy-5-sulfonatooxy-1-benzofuran-2-yl)methoxy]-2-methyl-1-benzofuran-6-yl] sulfate |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
Sodium;3-[(3-ethoxycarbonyl-6-methoxy-2-methyl-1-benzofuran-5-yl)oxymethyl]benzenesulfonate |
NA |
134000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
Disodium;[3-[(3-ethoxycarbonyl-2-methyl-5-sulfonatooxy-1-benzofuran-6-yl)oxymethyl]phenyl] sulfate |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
Disodium;[3-[[3-ethoxycarbonyl-5-[(3-ethoxycarbonyl-6-methoxy-5-sulfonatooxy-1-benzofuran-2-yl)methoxy]-2-methyl-1-benzofuran-6-yl]oxy]phenyl] sulfate |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
Sodium;[3-ethoxycarbonyl-2-methyl-6-[(3-propan-2-yloxyphenyl)methoxy]-1-benzofuran-5-yl] sulfate |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
Sodium;(3-ethoxycarbonyl-2-methyl-6-phenylmethoxy-1-benzofuran-5-yl) sulfate |
NA |
134000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
Sodium;(6-methoxy-2-methyl-3-phenylmethoxycarbonyl-1-benzofuran-5-yl) sulfate |
NA |
168000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
Sodium;[3-ethoxycarbonyl-6-[[3-(methoxymethoxy)phenyl]methoxy]-2-methyl-1-benzofuran-5-yl] sulfate |
NA |
229000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
Sodium;[6-(cyclohexylmethoxy)-3-ethoxycarbonyl-2-methyl-1-benzofuran-5-yl] sulfate |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
Dihydrospumigin N |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
Disodium;2-(6-methoxy-2-methyl-5-sulfonatooxy-1-benzofuran-3-carbonyl)oxyethyl sulfate |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |