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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
F2 Sodium;[3-ethoxycarbonyl-2-methyl-6-[(4-propan-2-yloxyphenyl)methoxy]-1-benzofuran-5-yl] sulfate NA 500000 NA NA NA NA TTD
F2 Disodium;2-methyl-6-phenylmethoxy-5-sulfonatooxy-1-benzofuran-3-carboxylate NA 500000 NA NA NA NA TTD
F2 Sodium;3-[(3-ethoxycarbonyl-2-methyl-6-phenylmethoxy-1-benzofuran-5-yl)oxymethyl]benzenesulfonate NA 500000 NA NA NA NA TTD
F2 Disodium;3-[[3-methoxycarbonyl-2-methyl-6-[(3-sulfonatooxyphenyl)methoxy]-1-benzofuran-5-yl]oxymethyl]benzenesulfonate NA 500000 NA NA NA NA TTD
F2 N-[3-(2-Amino-ethoxy)-5-methyl-phenyl]-benzenesulfonamide 240000 NA NA NA NA NA TTD
F2 2-[3-[3-(4-Benzylpiperidine-1-carbonyl)-5-chlorophenoxy]propoxy]guanidine 1500000 NA NA NA NA NA TTD
F2 acetic acid;(2S)-N-[(4-carbamimidoylphenyl)methyl]-1-ethylsulfonylpyrrolidine-2-carboxamide 117000 NA NA NA NA NA TTD
F2 5-[[(2S)-1-amino-4-methyl-1-oxopentan-2-yl]carbamoyl]-2-[2-[[4-(aminomethyl)phenyl]carbamoyl]-4-(methylamino)phenyl]benzoic acid NA 200000 NA NA NA NA TTD
F2 (2S)-N-[(1S)-1-{[(2S)-5-carbamimidamido-1-oxo-1-(1,3-thiazol-2-yl)pentan-2-yl]carbamoyl}-2-methylpropyl]-2-acetamido-4-methylpentanamide NA 200000 NA NA NA NA TTD
F2 H-Pro-Glu-His-Pro-Ala-Glu-Thr-Glu-Tyr-Asp-Ser-Leu-Tyr-Pro-Glu-Asp-Asp-Leu-OH NA 130000 NA NA NA NA TTD
F2 Benzamidine HCl hydrate 1000000 NA NA NA NA NA TTD
F2 Amiloride NA 250000 NA NA NA NA PubChem
F2 [2-[(3,5-Dimethyl-1-phenylpyrazol-4-yl)amino]-2-oxoethyl] 2-(2-oxo-1,3-benzoxazol-3-yl)acetate NA 200000 NA NA NA NA TTD
F2 [2-[(3,5-Dimethyl-1-phenylpyrazol-4-yl)amino]-2-oxoethyl] 2-phenylacetate NA 200000 NA NA NA NA TTD
F2 [2-[(3,5-Dimethyl-1-phenylpyrazol-4-yl)amino]-2-oxoethyl] 2-(4-oxoquinazolin-3-yl)acetate NA 200000 NA NA NA NA TTD
F2 Diphenyl 1-(methylsulfonylamino)-2-(4-guanidinophenyl)-ethanephosphonate NA 125000 NA NA NA NA TTD
F2 Dalfampridine 2000000 NA NA NA NA NA PubChem|TTD
F2 4-(2-Hydroxyethylamino)-pyridine 500000 NA NA NA NA NA TTD
F2 N-[2-(3-Carbamimidoyl-phenoxy)-ethyl]-4-[1-(1-imino-ethyl)-piperidin-4-yloxy]-benzamide 440000 NA NA NA NA NA TTD
F2 2-[3-[3-Chloro-5-(4-phenylpiperazine-1-carbonyl)phenoxy]propoxy]guanidine 2900000 NA NA NA NA NA TTD