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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
F2 [4-[[4-[[4-(Diaminomethylideneamino)phenyl]methylcarbamoyl]piperazine-1-carbonyl]oxymethyl]cyclohexyl]methyl 4-[[4-(diaminomethylideneamino)phenyl]methylcarbamoyl]piperazine-1-carboxylate 1000000 NA NA NA NA NA TTD
F2 [5-[4-[2-(1-Carbamimidoylpiperidin-4-yl)acetyl]piperazine-1-carbonyl]oxycyclooctyl] 4-[2-(1-carbamimidoylpiperidin-4-yl)acetyl]piperazine-1-carboxylate 130000 NA NA NA NA NA TTD
F2 [5-[4-[2-(1-Carbamimidoylpiperidin-4-yl)ethylcarbamoyl]piperazine-1-carbonyl]oxycyclooctyl] 4-[2-(1-carbamimidoylpiperidin-4-yl)ethylcarbamoyl]piperazine-1-carboxylate 112000 NA NA NA NA NA TTD
F2 [5-[4-[3-(1-Carbamimidoylpiperidin-4-yl)propanoyl]piperazine-1-carbonyl]oxycyclooctyl] 4-[3-(1-carbamimidoylpiperidin-4-yl)propanoyl]piperazine-1-carboxylate 213000 NA NA NA NA NA TTD
F2 [5-[4-[3-[4-(Diaminomethylideneamino)phenyl]propanoyl]piperazine-1-carbonyl]oxycyclooctyl] 4-[3-[4-(diaminomethylideneamino)phenyl]propanoyl]piperazine-1-carboxylate 537000 NA NA NA NA NA TTD
F2 [5-[4-[2-[4-(2-Aminoethyl)phenyl]acetyl]piperazine-1-carbonyl]oxycyclooctyl] 4-[2-[4-(2-aminoethyl)phenyl]acetyl]piperazine-1-carboxylate 1000000 NA NA NA NA NA TTD
F2 [5-[4-(4-Aminobutylcarbamoyl)piperazine-1-carbonyl]oxycyclooctyl] 4-(4-aminobutylcarbamoyl)piperazine-1-carboxylate 1000000 NA NA NA NA NA TTD
F2 [5-[4-[[4-(Aminomethyl)phenyl]methylcarbamoyl]piperazine-1-carbonyl]oxycyclooctyl] 4-[[4-(aminomethyl)phenyl]methylcarbamoyl]piperazine-1-carboxylate 1000000 NA NA NA NA NA TTD
F2 [5-[4-[2-[4-(Diaminomethylideneamino)phenyl]acetyl]piperazine-1-carbonyl]oxycyclooctyl] 4-[2-[4-(diaminomethylideneamino)phenyl]acetyl]piperazine-1-carboxylate 255000 NA NA NA NA NA TTD
F2 [5-[4-(5-Aminopentylcarbamoyl)piperazine-1-carbonyl]oxycyclooctyl] 4-(5-aminopentylcarbamoyl)piperazine-1-carboxylate 1000000 NA NA NA NA NA TTD
F2 [5-[4-(6-Aminohexylcarbamoyl)piperazine-1-carbonyl]oxycyclooctyl] 4-(6-aminohexylcarbamoyl)piperazine-1-carboxylate 1000000 NA NA NA NA NA TTD
F2 [5-[4-[[4-(Diaminomethylideneamino)phenyl]methylcarbamoyl]piperazine-1-carbonyl]oxycyclooctyl] 4-(5-aminopentylcarbamoyl)piperazine-1-carboxylate 1000000 NA NA NA NA NA TTD
F2 [5-[4-[(1-Carbamimidoylpiperidin-4-yl)methylcarbamoyl]piperazine-1-carbonyl]oxycyclooctyl] 4-[(1-carbamimidoylpiperidin-4-yl)methylcarbamoyl]piperazine-1-carboxylate 146000 NA NA NA NA NA TTD
F2 N-[(2S)-1-(4-methylpiperidin-1-yl)-1-oxo-5-(pyrimidin-2-ylamino)pentan-2-yl]naphthalene-2-sulfonamide NA 115000 NA NA NA NA TTD
F2 Piperidine-1-carboximidamide 111000|NA NA NA|107000|197000 NA NA NA ChEMBL|PubChem
F2 3-(Benzylsulfamoyl)benzenecarboximidamide 102000 NA NA NA NA NA TTD
F2 [5-[4-[[4-(Diaminomethylideneamino)phenyl]methylcarbamoyl]piperazine-1-carbonyl]oxycyclooctyl] 4-(4-aminobutylcarbamoyl)piperazine-1-carboxylate 1000000 NA NA NA NA NA TTD
F2 [5-[4-[[4-(Diaminomethylideneamino)phenyl]methylcarbamoyl]piperazine-1-carbonyl]oxycyclooctyl] 4-(3-aminopropylcarbamoyl)piperazine-1-carboxylate 1000000 NA NA NA NA NA TTD
F2 [4-[[4-[[4-(Diaminomethylideneamino)phenyl]methylcarbamoyl]piperazine-1-carbonyl]oxymethyl]-1-bicyclo[2.2.2]octanyl]methyl 4-[[4-(diaminomethylideneamino)phenyl]methylcarbamoyl]piperazine-1-carboxylate 123000 NA NA NA NA NA TTD
F2 Beta-Sitosterol NA 1500000 NA NA NA NA PubChem