| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| F2 |
2-(2,6-Difluoro-phenyl)-7-nitro-benzo[d][1,3]oxazin-4-one |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
{[2-(4-Carbamimidoyl-benzylcarbamoyl)-cyclopentanecarbonyl]-amino}-phenyl-acetic acid |
NA |
132000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
5-chloropyridin-3-yl 6-(chloromethyl)-2-oxo-2H-chromene-3-carboxylate |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
3-[Bis-(6-amino-hexyl)-amino]-tetrahydro-thiopyran-4-one |
10000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(+) Cyclopentane-1,2-dicarboxylic acid 1-benzylamide 2-(4-carbamimidoyl-benzylamide) |
NA |
132000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
4-[5-Carbamimidoyl-2-(2-carboxy-2-oxo-ethyl)-phenoxy]-3-{4-[1-(1-imino-ethyl)-piperidin-4-yloxy]-benzoylamino}-butyric acid |
540000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
3-(4-Carbamimidoyl-benzoylamino)-4-(3-carbamimidoyl-phenoxy)-butyric acid |
1500000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(3R)-4-[5-carbamimidoyl-2-(2-carboxy-2-oxoethyl)phenoxy]-3-[(1-pyridin-4-ylpiperidine-4-carbonyl)amino]butanoic acid |
680000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
3-[4-Carbamimidoyl-2-[2-[(1-pyridin-4-ylpiperidine-4-carbonyl)amino]ethoxy]phenyl]-2-oxopropanoic acid |
140000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
2-Phenyl-1H-benzoimidazole-5-carboxamidine |
340000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
N-[2-(3-Carbamimidoyl-phenoxy)-ethyl]-4-(pyrrolidine-1-carbonyl)-benzamide |
110000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(3S)-3-[(4-carbamimidoylbenzoyl)amino]-4-(3-carbamimidoylphenoxy)butanoic acid |
1500000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
Cyclohex-2-ene-1,2-dicarboxylic acid 1-(4-carbamimidoyl-benzylamide) 2-cyclohexylamide |
NA |
130000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
Cyclohex-2-ene-1,2-dicarboxylic acid 1-(4-carbamimidoyl-benzylamide) 2-phenylamide |
NA |
130000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
{[2-(4-Carbamimidoyl-benzylcarbamoyl)-cyclopent-1-enecarbonyl]-o-tolyl-amino}-acetic acid |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
Cyclohex-2-ene-1,2-dicarboxylic acid 2-benzylamide 1-(4-carbamimidoyl-benzylamide) |
NA |
109000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
4-Acetyl-1-[1-(5-dimethylamino-naphthalene-1-sulfonyl)-pyrrolidine-2-carbonyl]-6-methyl-hexahydro-cyclopenta[b]pyrrol-5-one |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
2-(2,3-Dihydro-indole-1-carbonyl)-cyclopent-1-enecarboxylic acid 4-carbamimidoyl-benzylamide |
NA |
130000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
[4-(6-Chloro-naphthalene-2-sulfonyl)-piperazin-1-yl]-(5-methyl-4,5,6,7-tetrahydro-thiazolo[5,4-c]pyridin-2-yl)-methanone |
NA |
560000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
1,4,7-Tribenzyl-1,4,7-triazonane |
410000 |
NA |
NA |
NA |
NA |
NA |
TTD |