| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| JAK2 |
US10040781, Example 619 |
NA |
364000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
US10040781, Example 545 |
NA |
659000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
US10040781, Example 416 |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
US10040781, Example 588 |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
2-(((3R,4S)-1-(3-cyanopropanoyl)-3-fluoropiperidin-4-yl)oxy)-5-(4-((4-(4-(oxetan-3-yl)piperazin-1-yl)phenyl)amino)-1,3,5-triazin-2-yl)benzonitrile |
NA |
694000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
(R)-2-((1-(2,2-difluoroacetyl)pyrrolidin-3-yl)oxy)-5-(4-((4-(4-(oxetan-3-yl)piperazin-1-yl)phenyl)amino)-1,3,5-triazin-2-yl)benzonitrile |
NA |
560000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
US10040781, Example 614 |
NA |
268000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
2-(((3R,4S)-3-fluoro-1-(pyridin-2-yl)piperidin-4-yl)oxy)-5-(4-((4-(4-(oxetan-3-yl)piperazin-1-yl)phenyl)amino)-1,3,5-triazin-2-yl)benzonitrile |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
2-(((2R,4S)-1-((S)-2-hydroxypropanoyl)-2-methylpiperidin-4-yl)oxy)-5-(4-((4-(4-(oxetan-3-yl)piperazin-1-yl)phenyl)amino)-1,3,5-triazin-2-yl)benzonitrile |
NA |
593000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
US10040781, Example 352 |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
US10040781, Example 618 |
NA |
162000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
2-((4,4-Difluoropyrrolidin-3-yl)oxy)-5-(4-((4-(4-(oxetan-3-yl)piperazin-1-yl)phenyl)amino)-1,3,5-triazin-2-yl)benzonitrile |
NA |
308000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
5-(4-((1-(difluoromethyl)-1H-pyrazol-4-yl)amino)-1,3,5-triazin-2-yl)-2-(((3R,4S)-3-fluoropiperidin-4-yl)oxy)benzonitrile |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
US10040781, Example 590 |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
US10040781, Example 227 |
NA |
333000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
5-(4-((3-(2-hydroxypropan-2-yl)phenyl)amino)-1,3,5-triazin-2-yl)-2-((tetrahydro-2H-pyran-4-yl)oxy)benzonitrile |
NA |
811000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
US10040781, Example 549 |
NA |
179000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
US10040781, Example 481 |
NA |
320000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
US10040781, Example 540 |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
US10040781, Example 406 |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB |