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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
PPARG Clofibric Acid NA NA NA 309000|300000 NA NA BindingDB|PubChem|TTD
PPARG Valproic Acid NA NA NA NA 794328 NA PubChem
PPARG Cefazolin NA NA NA NA NA 300000 PubChem
PPARG Fenofibrate NA NA NA 300000 NA NA BindingDB|PubChem
PPARG Gemfibrozil NA NA NA 147800 NA NA BindingDB|PubChem|TTD
PPARG Bezafibrate NA NA NA 137000 NA NA PubChem
PPARG Meropenem NA NA NA NA NA 300000 PubChem
PPARG methyl 2-(5-(2-(2-(biphenyl-4-yl)-5-methyloxazol-4-yl)ethoxy)-1-(4-chlorobenzoyl)-2-methyl-1H-indol-3-yl)acetate NA NA NA 20000000 NA NA BindingDB|TTD
PPARG (2S)-2-(4-benzoylanilino)-3-(4-phenylmethoxyphenyl)propanoic acid 169000000 NA NA NA NA NA BindingDB
PPARG (2S)-2-(2-benzoylanilino)-3-(4-phenylmethoxyphenyl)propanoic acid 164000000 NA NA NA NA NA BindingDB
PPARG Oleic Acid NA NA NA NA NA 300000 PubChem
PPARG 1-[4-[2-(Benzenesulfonamido)ethyl]phenyl]sulfonyl-3-(4-methoxyphenyl)thiourea NA 1000000 NA NA NA NA BindingDB|TTD
PPARG Mycophenolic Acid NA NA 110000 NA NA NA BindingDB|PubChem
PPARG 3-(((6-((5-Cyclopropyl-3-(2,6-dichlorophenyl)isoxazol-4-yl)methoxy)-2-(trifluoromethyl)pyridin-3-yl)(methyl)amino)methyl)benzoic acid NA NA NA 1450000 NA NA BindingDB|TTD
PPARG 3-(2,3,10,11-Tetramethoxy-1,4-dihydroisoquinolino[2,1-b]isoquinolin-7-ium-8-yl)propanoic acid NA NA NA 220000 NA NA BindingDB|TTD
PPARG (2S)-2-(4-oxopentan-2-ylideneamino)-3-(4-phenylmethoxyphenyl)propanoic acid 175000000 NA NA NA NA NA BindingDB
PPARG [3H]rosiglitazone NA NA NA 10000000 NA NA BindingDB
PPARG 2-[2-[Diazenyl(phenyl)methyl]anilino]-3-[4-[2-[methyl(pyridin-2-yl)amino]ethoxy]phenyl]propanoic acid 144000000 NA NA NA NA NA BindingDB
PPARG methyl (2S)-2-[(4-oxo-4-phenylbutan-2-ylidene)amino]-3-(4-phenylmethoxyphenyl)propanoate 163000000 NA NA NA NA NA BindingDB
PPARG (2S)-2-[(4-oxo-4-phenylbutan-2-ylidene)amino]-3-(4-phenylmethoxyphenyl)propanoic acid 126000000 NA NA NA NA NA BindingDB