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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
PPARG methyl 2-(1-(4-chlorobenzoyl)-2-methyl-5-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)-1H-indol-3-yl)acetate NA NA NA 620000000 NA NA BindingDB|TTD
PPARG 2-(5-(2-(2-(biphenyl-4-yl)-5-methyloxazol-4-yl)ethoxy)-1-(4-chlorobenzoyl)-2-methyl-1H-indol-3-yl)acetic acid NA NA NA 40000000 NA NA BindingDB|TTD
PPARG 2-(4-(Benzyloxy)-2-(2,6-dichlorophenylamino)phenyl)acetic acid NA NA NA 6030000000 NA NA BindingDB
PPARG 2-(1-(4-chlorobenzoyl)-2-methyl-5-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)-1H-indol-3-yl)acetic acid NA NA NA 1230000000 NA NA BindingDB
PPARG (2S)-3-[4-[2-[1,3-benzoxazol-2-yl(methyl)amino]ethoxy]phenyl]-2-(2-phenoxyanilino)propanoic acid 118000000|118850222.7 NA NA NA NA|NA NA|NA BindingDB|TTD
PPARG Cefepime NA NA NA NA NA 300000|200000 PubChem
PPARG Ceftazidime NA NA NA NA NA 300000 PubChem
PPARG Aztreonam NA NA NA NA NA 400000 PubChem
PPARG Mifobate NA 140000 NA NA NA NA BindingDB|TTD
PPARG Fenofibric Acid NA NA|744000 NA 217000|300000|NA NA NA BindingDB|PubChem
PPARG GW 1929 113000000 NA NA NA NA NA BindingDB
PPARG Carumonam NA NA NA NA NA 500000 PubChem
PPARG 2-Phenylphenol NA NA NA NA 316228 NA PubChem
PPARG Doripenem NA NA NA NA NA 300000 PubChem
PPARG 2,4-Dimethylphenol NA NA NA NA 1412540 NA PubChem
PPARG Rosiglitazone NA NA NA 191500|10000000 NA NA BindingDB|PubChem
PPARG (2S)-2-[(4-oxo-4-phenylbutan-2-ylidene)amino]-3-(4-phenylmethoxyphenyl)propanamide 170000000 NA NA NA NA NA BindingDB
PPARG (2S)-5-(4-methoxyanilino)-2-[(4-methylphenyl)sulfonylamino]-5-oxopentanoic acid NA 275000 NA NA NA NA BindingDB
PPARG (2S)-5-anilino-2-[(4-methylphenyl)sulfonylamino]-5-oxopentanoic acid NA 140000 NA NA NA NA BindingDB
PPARG 3-((Amino(imino)methyl)hydrazono)-N-(2,4-dimethylphenyl)butanamide NA 180000 NA NA NA NA BindingDB