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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
PPIA 1-(m-tolyl)-3-(3-oxo-1H-isobenzofuran-5-yl)thiourea NA NA 141000 NA NA NA BindingDB
PPIA 1-(4-Methoxyphenyl)-3-(3-oxo-1,3-dihydroisobenzofuran-5-yl)thiourea NA NA 171800 NA NA NA BindingDB
PPIA 1-(4-Chlorophenyl)-3-(3-oxo-1,3-dihydroisobenzofuran-5-yl)thiourea NA NA 222200 NA NA NA BindingDB
PPIA 1-(4-Fluorophenyl)-3-(3-oxo-1,3-dihydroisobenzofuran-5-yl)thiourea NA NA 227300 NA NA NA BindingDB
PPIA Ac-Val-Gln-Ala-Gly-Pro-D-Ile-D-Ala-NH2 NA 2500000 NA NA NA NA BindingDB|TTD
PPIA Ac-Val-His-Ala-Gly-Pro-D-Ile-D-Ala-NH2 NA 850000 NA NA NA NA BindingDB|TTD
PPIA 4-[[(2S)-1-[2-[[(2S)-2-[[(2S)-2-[[(2S)-2-acetamido-3-methylbutanoyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]propanoyl]amino]acetyl]pyrrolidine-2-carbonyl]amino]-N-[(2R)-1-amino-1-oxopropan-2-yl]piperidine-4-carboxamide NA 10000000 NA NA NA NA TTD
PPIA Ac-Val-His-Ala-Gly-Pro-Aib-D-Ala-NH2 NA 10000000 NA NA NA NA TTD
PPIA Ac-Val-His-Ala-Gly-Pro-Gly-D-Ala-NH2 NA 2800000 NA NA NA NA BindingDB|TTD
PPIA Ac-Val-His-Aib-Gly-Pro-D-Ile-D-Ala-NH2 NA 760000 NA NA NA NA BindingDB|TTD
PPIA Ac-Val-His-Ala-Gly-Pro-Gln-D-Ala-NH2 NA 1300000 NA NA NA NA BindingDB|TTD
PPIA Ac-Val-His-Ala-Gly-Pro-Val-D-Ala-NH2 NA 1500000 NA NA NA NA BindingDB|TTD
PPIA Ac-Val-His-Ala-Gly-Pro-D-Phg-D-Ala-NH2 NA 970000 NA NA NA NA BindingDB|TTD
PPIA Ac-Val-His-Ala-Gly-Pro-Phg-D-Ala-NH2 NA 820000 NA NA NA NA BindingDB|TTD
PPIA 6-Benzyl-6-benzyloxycarbonylamino-5-oxo-hexahydro-indolizine-8a-carboxylic acid methyl ester NA NA 124000 NA NA NA BindingDB
PPIA Ac-Val-His-Ala-Gly-D-Pro-Val-Ala-NH2 NA 1500000 NA NA NA NA BindingDB|TTD
PPIA Ac-Val-Gln-Ala-Gly-D-Pro-Ile-Ala-NH2 NA 2500000 NA NA NA NA BindingDB|TTD
PPIA deamino-His-Ala-Gly-D-Pro-Ile-Ala-NH2 NA 2600000 NA NA NA NA BindingDB|TTD
PPIA isovaleryl-His-Ala-Gly-D-Pro-Ile-Ala-NH2 NA 165000 NA NA NA NA BindingDB|TTD
PPIA Ac-Val-His-Ala-Gly-D-Pro-Ile-Ala-NH2 NA 850000 NA NA NA NA BindingDB|TTD