| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PPARG |
Phenol |
NA |
NA |
NA |
NA |
1122020 |
NA |
PubChem |
| PPIA |
Ac-Val-His-Ala-Gly-Pro-Ile-NHbenzhydryl |
NA |
1500000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PPIA |
6-Benzyl-6-tert-butoxycarbonylamino-5-oxo-hexahydro-indolizine-8a-carboxylic acid methyl ester |
NA |
NA |
140000 |
NA |
NA |
NA |
BindingDB |
| PPIA |
(6R,15S,18S)-6-amino-6-methyl-2,5,17-trioxo-8,13-dioxa-1,4,16-triazabicyclo[16.3.0]henicosane-15-carboxylic acid;2,2,2-trifluoroacetic acid |
NA |
NA |
127000 |
NA |
NA |
NA |
BindingDB |
| PPIA |
(6R,15S,18S)-6-(cyclobutanecarbonylamino)-6-methyl-2,5,17-trioxo-8,13-dioxa-1,4,16-triazabicyclo[16.3.0]henicosane-15-carboxylic acid |
NA |
NA |
139000 |
NA |
NA |
NA |
BindingDB |
| PPIA |
Ethyl 2-[[(4-aminophenyl)methyl-[(1-methyl-1,2,3-triazol-4-yl)methyl]carbamoyl]amino]ethanoate |
NA |
NA |
135000 |
NA |
NA |
NA |
BindingDB |
| PPIA |
Ethyl 2-[[(4-aminophenyl)methyl-ethylcarbamoyl]amino]acetate |
NA |
NA |
200000 |
NA |
NA |
NA |
BindingDB |
| PPIA |
ethyl 2-[[(4-aminophenyl)methyl-(1~{H}-1,2,3,4-tetrazol-5-ylmethyl)carbamoyl]amino]ethanoate |
NA |
NA |
139000 |
NA |
NA |
NA |
BindingDB |
| PPIA |
Ethyl 2-[[(4-aminophenyl)methyl-propyl-carbamoyl]amino]ethanoate |
NA |
NA |
266000 |
NA |
NA |
NA |
BindingDB |
| PPIA |
Ethyl 2-[[(4-aminophenyl)methyl-[(2-methyl-1,2,3,4-tetrazol-5-yl)methyl]carbamoyl]amino]ethanoate |
NA |
NA |
184000 |
NA |
NA |
NA |
BindingDB |
| PPIA |
1-[4-[(5-Methylisoxazol-3-yl)sulfamoyl]phenyl]-3-(p-tolyl)thiourea |
NA |
NA |
118800 |
NA |
NA |
NA |
BindingDB |
| PPIA |
4-(3-(4-Fluorophenyl)thioureido)-N-(5-methylisoxazol-3-yl)benzenesulfonamide |
NA |
NA |
109500 |
NA |
NA |
NA |
BindingDB |
| PPIA |
Ethyl 2-[[(4-aminophenyl)methyl-(cyanomethyl)carbamoyl]amino]acetate |
NA |
NA |
990000 |
NA |
NA |
NA |
BindingDB |
| PPIA |
ethyl 2-[[ethyl-[[(1R,9R,10S)-10-hydroxy-12-oxa-8-azatricyclo[7.3.1.02,7]trideca-2(7),3,5-trien-4-yl]methyl]carbamoyl]amino]acetate |
NA |
NA |
700000 |
NA |
NA |
NA |
BindingDB |
| PPIA |
1-(4-Methoxyphenyl)-3-(naphthalen-2-yl)thiourea |
NA |
NA |
124400 |
NA |
NA |
NA |
BindingDB |
| PPIA |
4-(3-(4-Chlorophenyl)thioureido)-N-(5-methylisoxazol-3-yl)benzenesulfonamide |
NA |
NA |
107300 |
NA |
NA |
NA |
BindingDB |
| PPIA |
4-(3-(4-Methoxyphenyl)thioureido)-N-(5-methylisoxazol-3-yl)benzenesulfonamide |
NA |
NA |
100700 |
NA |
NA |
NA |
BindingDB |
| PPIA |
1-(3-Bromophenyl)-3-(3-oxo-1,3-dihydroisobenzofuran-5-yl)thiourea |
NA |
NA |
125100 |
NA |
NA |
NA |
BindingDB |
| PPIA |
1-(3-Chlorophenyl)-3-(3-oxo-1,3-dihydroisobenzofuran-5-yl)thiourea |
NA |
NA |
133300 |
NA |
NA |
NA |
BindingDB |
| PPIA |
1-(3,5-Difluorophenyl)-3-(3-oxo-1,3-dihydroisobenzofuran-5-yl)thiourea |
NA |
NA |
512800 |
NA |
NA |
NA |
BindingDB |