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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
ABCG2 1-(2-Aminophenyl)-3-(4-(2-(3,4-dihydroisoquinolin-2(1H)-yl)ethyl)phenyl)urea NA 102000 NA NA NA NA BindingDB
ABCG2 Amphotericin B NA 127000 NA NA NA NA PubChem
ABCG2 Novobiocin NA 104000 NA NA NA NA PubChem|TTD
ABCG2 5-[(4-bromophenyl)methoxy]-N-[2-(5-methoxy-1H-indol-3-yl)ethyl]-4-oxochromene-2-carboxamide NA NA NA 130016958 NA NA BindingDB
ABCG2 Progesterone NA 125892.54|125893 NA NA NA NA BindingDB|PubChem|TTD
ABCG2 Proguanil NA 118000 NA NA NA NA BindingDB|PubChem
ABCG2 Amprenavir NA 181000 NA NA NA NA BindingDB|PubChem
ABCG2 Dexverapamil NA 524807 NA NA NA NA BindingDB
ABCG2 [(3R,4S,5S,6S)-5-hydroxy-6-[4-hydroxy-3-[[4-hydroxy-3-(3-methylbut-2-enyl)benzoyl]amino]-8-methyl-2-oxochromen-7-yl]oxy-3-methoxy-2,2-dimethyloxan-4-yl] carbamate NA 104000 NA NA NA NA BindingDB
ABCG2 5-[(4-bromophenyl)methoxy]-N-[2-(1-methylindol-3-yl)ethyl]-4-oxochromene-2-carboxamide NA NA NA 299916252 NA NA BindingDB
ABCG2 5-[(4-bromophenyl)methoxy]-N-[2-(1H-indol-3-yl)ethyl]-N-methyl-4-oxochromene-2-carboxamide NA NA NA 1109174815 NA NA BindingDB
ABCG2 5-[(4-bromophenyl)methoxy]-N-[2-(5-methoxy-1H-indol-3-yl)ethyl]-N-methyl-4-oxochromene-2-carboxamide NA NA NA 959400632 NA NA BindingDB
ABCG2 6-[(4-bromophenyl)methoxy]-N-[2-(5-methoxy-1H-indol-3-yl)ethyl]-4-oxochromene-2-carboxamide NA NA NA 289734359 NA NA BindingDB
ABCG2 6-[(4-bromophenyl)methoxy]-N-[2-(1H-indol-3-yl)ethyl]-N-methyl-4-oxochromene-2-carboxamide NA NA NA 2582260191 NA NA BindingDB
ABCG2 6-[(4-bromophenyl)methoxy]-N-methyl-N-[2-(1-methylindol-3-yl)ethyl]-4-oxochromene-2-carboxamide NA NA NA 2060629913 NA NA BindingDB
ABCG2 5-[(4-bromophenyl)methoxy]-N-[2-(6-methoxy-1H-indol-3-yl)ethyl]-4-oxochromene-2-carboxamide NA NA NA 100000000 NA NA BindingDB
ABCG2 5-[(4-bromophenyl)methoxy]-N-methyl-N-[2-(1-methylindol-3-yl)ethyl]-4-oxochromene-2-carboxamide NA NA NA 1000000000 NA NA BindingDB
ABCG2 7-[(4-bromophenyl)methoxy]-N-[2-(5-methoxy-1H-indol-3-yl)ethyl]-4-oxochromene-2-carboxamide NA NA NA 1270574105 NA NA BindingDB
ABL1 1H-Pyrrole-3-carboxamide, 5-((5-fluoro-1,2-dihydro-2-oxo-3H-indol-3-ylidene)methyl)-N-((2S)-2-hydroxy-3-(4-morpholinyl)propyl)-2,4-dimethyl- NA NA 2100000 NA NA NA BindingDB
ABL1 Raf-265 NA NA 580000 NA NA NA BindingDB