| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| ACHE |
|
NA |
970000 |
NA |
NA |
NA |
NA |
BindingDB |
| ACHE |
|
NA |
1660000 |
NA |
NA |
NA |
NA |
BindingDB |
| ACHE |
|
NA |
2270000 |
NA |
NA |
NA |
NA |
BindingDB |
| ACHE |
|
NA |
2490000 |
NA |
NA |
NA |
NA |
BindingDB |
| ACHE |
3-[(1S)-1-(4-fluorophenyl)-5-(5-phenyl-1H-1,2,4-triazol-3-yl)-3H-2-benzofuran-1-yl]-N,N-dimethylpropan-1-amine |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| ACHE |
2-[3-[(1S)-1-[3-(dimethylamino)propyl]-1-(4-fluorophenyl)-3H-2-benzofuran-5-yl]-1H-1,2,4-triazol-5-yl]aniline |
NA |
359720 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ACHE |
3-[5-[(1S)-1-[3-(dimethylamino)propyl]-1-(4-fluorophenyl)-3H-2-benzofuran-5-yl]-1H-1,2,4-triazol-3-yl]aniline |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| ACHE |
|
NA |
387560 |
NA |
NA |
NA |
NA |
BindingDB |
| ACHE |
3-[(1S)-1-(4-fluorophenyl)-5-[3-(3-nitrophenyl)-1H-1,2,4-triazol-5-yl]-3H-2-benzofuran-1-yl]-N,N-dimethylpropan-1-amine |
NA |
138230 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ACHE |
3-[(1S)-1-(4-fluorophenyl)-5-[3-(3-methylphenyl)-1H-1,2,4-triazol-5-yl]-3H-2-benzofuran-1-yl]-N,N-dimethylpropan-1-amine |
NA |
133230 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ACHE |
3-[(1S)-5-[3-(3-chlorophenyl)-1H-1,2,4-triazol-5-yl]-1-(4-fluorophenyl)-3H-2-benzofuran-1-yl]-N,N-dimethylpropan-1-amine |
NA |
412560 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ACHE |
3-[(1S)-1-(4-fluorophenyl)-5-[5-(2-fluorophenyl)-1H-1,2,4-triazol-3-yl]-3H-2-benzofuran-1-yl]-N,N-dimethylpropan-1-amine |
NA |
187510 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ACHE |
3-[(1S)-1-(4-fluorophenyl)-5-[5-(4-fluorophenyl)-1H-1,2,4-triazol-3-yl]-3H-2-benzofuran-1-yl]-N,N-dimethylpropan-1-amine |
NA |
260630 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ACHE |
3-[(1S)-1-(4-fluorophenyl)-5-[5-(2-iodophenyl)-1H-1,2,4-triazol-3-yl]-3H-2-benzofuran-1-yl]-N,N-dimethylpropan-1-amine |
NA |
310310 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ACHE |
3-[(1S)-1-(4-fluorophenyl)-5-[3-(3-iodophenyl)-1H-1,2,4-triazol-5-yl]-3H-2-benzofuran-1-yl]-N,N-dimethylpropan-1-amine |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| ACHE |
3-[(1S)-1-(4-fluorophenyl)-5-[5-(4-iodophenyl)-1H-1,2,4-triazol-3-yl]-3H-2-benzofuran-1-yl]-N,N-dimethylpropan-1-amine |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| ACHE |
3-[(1S)-1-(4-fluorophenyl)-5-[5-(2-methoxyphenyl)-1H-1,2,4-triazol-3-yl]-3H-2-benzofuran-1-yl]-N,N-dimethylpropan-1-amine |
NA |
161340 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ACHE |
3-[(1S)-1-(4-fluorophenyl)-5-[3-(3-methoxyphenyl)-1H-1,2,4-triazol-5-yl]-3H-2-benzofuran-1-yl]-N,N-dimethylpropan-1-amine |
NA |
123770 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ACHE |
3-[(1S)-1-(4-fluorophenyl)-5-[5-[4-(2H-tetrazol-5-yl)phenyl]-1H-1,2,4-triazol-3-yl]-3H-2-benzofuran-1-yl]-N,N-dimethylpropan-1-amine |
NA |
251670 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ACHE |
Ethopropazine Hydrochloride |
NA|12100000 |
1020000|NA |
NA |
NA |
NA |
NA |
PubChem |