| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| ACHE |
1-[3-[4-(4-Ethylpiperazin-1-yl)phenyl]-5-(4-methoxyphenyl)-3,4-dihydropyrazol-2-yl]ethanone |
NA |
221200 |
NA |
NA |
NA |
NA |
TTD |
| ACHE |
1-[5-(3,6-dimethyl-2,4-dioxopyrimidin-1-yl)pentyl]-N-hydroxy-1,2,4-triazole-3-carboxamide |
NA |
NA |
5500000 |
NA |
NA |
NA |
BindingDB |
| ACHE |
4-(4-bromophenyl)-2-[(E)-2-phenylethenyl]-1,3-thiazole |
NA |
229999 |
NA |
NA |
NA |
NA |
BindingDB |
| ACHE |
[3-[2-(cyclohexylamino)-1-hydroxyethyl]phenyl] N,N-dimethylcarbamate;hydrochloride |
NA |
792000 |
NA |
NA |
NA |
NA |
BindingDB |
| ACHE |
[4-[2-(cyclohexylamino)-1-hydroxyethyl]phenyl] N,N-dimethylcarbamate;hydrochloride |
NA |
266000 |
NA |
NA |
NA |
NA |
BindingDB |
| ACHE |
Barbigerone |
NA |
121600 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ACHE |
Xylopine |
NA |
125900 |
NA |
NA |
NA |
NA |
BindingDB |
| ACHE |
(+)-(S)-ar-Turmerone |
NA |
191100 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ACHE |
3-[12-(Benzylmethylamino)dodecyloxy]xanthen-9-one |
NA |
908000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ACHE |
(-)-Corydalmine |
NA |
211200 |
NA |
NA |
NA |
NA |
BindingDB |
| ACHE |
2-[(E)-hydroxyiminomethyl]-4-methyl-6-[(4-pyridin-4-ylpiperazin-1-yl)methyl]phenol |
NA |
484000 |
NA |
NA |
NA |
NA |
BindingDB |
| ACHE |
4-chloro-2-[(E)-hydroxyiminomethyl]-6-[(4-pyrazol-1-ylanilino)methyl]phenol |
NA |
3035000 |
NA |
NA |
NA |
NA |
BindingDB |
| ACHE |
2-[(E)-hydroxyiminomethyl]-4-methyl-6-[[4-(1,2,4-triazol-1-ylmethyl)anilino]methyl]phenol |
NA |
3255000 |
NA |
NA |
NA |
NA |
BindingDB |
| ACHE |
4-chloro-2-[(E)-hydroxyiminomethyl]-6-[[(3-phenylmethoxypyridin-2-yl)amino]methyl]phenol |
NA |
826000 |
NA |
NA |
NA |
NA |
BindingDB |
| ACHE |
2-[[4-[[2-(1-hydroxycyclohexyl)-2-(4-methoxyphenyl)ethyl]-methylamino]anilino]methyl]-6-[(E)-hydroxyiminomethyl]-4-methylphenol |
NA |
1256000 |
NA |
NA |
NA |
NA |
BindingDB |
| ACHE |
4-[[2-hydroxy-3-[(E)-hydroxyiminomethyl]-5-methylphenyl]methylamino]-N-(1,3-thiazol-2-yl)benzenesulfonamide |
NA |
5149000 |
NA |
NA |
NA |
NA |
BindingDB |
| ACHE |
4-[4-[[5-chloro-2-hydroxy-3-[(E)-hydroxyiminomethyl]phenyl]methylamino]phenyl]morpholin-3-one |
NA |
4177000 |
NA |
NA |
NA |
NA |
BindingDB |
| ACHE |
4-chloro-2-[(E)-hydroxyiminomethyl]-6-[(4-pyridin-4-ylpiperazin-1-yl)methyl]phenol |
NA |
262000 |
NA |
NA |
NA |
NA |
BindingDB |
| ACHE |
4-chloro-2-[(3-fluoro-4-morpholin-4-ylanilino)methyl]-6-[(E)-hydroxyiminomethyl]phenol |
NA |
5917000 |
NA |
NA |
NA |
NA |
BindingDB |
| ACHE |
6-chloro-3-[1-[[5-chloro-2-hydroxy-3-[(E)-hydroxyiminomethyl]phenyl]methyl]piperidin-4-yl]-1H-benzimidazol-2-one |
NA |
4148000 |
NA |
NA |
NA |
NA |
BindingDB |