| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| ACHE |
1-[3-(4-Nitrophenyl)-5-(4-phenylphenyl)-3,4-dihydropyrazol-2-yl]ethanone |
NA |
1550000 |
NA |
NA |
NA |
NA |
BindingDB |
| ACHE |
(16S)-16-ethyl-5-methoxy-15-methyl-11-methylidene-9,15-diazatetracyclo[10.3.1.02,10.03,8]hexadeca-2(10),3(8),4,6-tetraene |
NA |
279000 |
NA |
NA |
NA |
NA |
BindingDB |
| ACHE |
1-[5-Naphthalen-1-yl-3-(4-phenylphenyl)-3,4-dihydropyrazol-2-yl]ethanone |
NA |
1010000 |
NA |
NA |
NA |
NA |
BindingDB |
| ACHE |
1-[5-(2,4-Dimethoxyphenyl)-3-(4-phenylphenyl)-3,4-dihydropyrazol-2-yl]ethanone |
NA |
1120000 |
NA |
NA |
NA |
NA |
BindingDB |
| ACHE |
1-[3-(4-Phenylphenyl)-5-(3,4,5-trimethoxyphenyl)-3,4-dihydropyrazol-2-yl]ethanone |
NA |
1940000 |
NA |
NA |
NA |
NA |
BindingDB |
| ACHE |
2-(Azepan-1-ylmethyl)-5-(8-hydroxyoctyl)phenol |
NA |
785000 |
NA |
NA |
NA |
NA |
BindingDB |
| ACHE |
(1aS,2S,3S,7bS)-2-hydroxy-6-[2-(3-hydroxy-4-methoxyphenyl)ethyl]-3-methoxy-1a,2,3,7b-tetrahydrooxireno[2,3-h]chromen-4-one |
NA |
441600 |
NA |
NA |
NA |
NA |
BindingDB |
| ACHE |
1-[5-(2,5-Dimethoxyphenyl)-3-(4-phenylphenyl)-3,4-dihydropyrazol-2-yl]ethanone |
NA |
1700000 |
NA |
NA |
NA |
NA |
BindingDB |
| ACHE |
5,8-dihydroxy-3-methoxy-3,4-dihydro-2H-naphthalen-1-one |
NA |
949000 |
NA |
NA |
NA |
NA |
BindingDB |
| ACHE |
1-[3-(2,5-Dimethoxyphenyl)-5-(4-phenylphenyl)-3,4-dihydropyrazol-2-yl]ethanone |
NA |
1420000 |
NA |
NA |
NA |
NA |
BindingDB |
| ACHE |
5-Hydroxy-1-[12-[(3-hydroxyphenyl)methyl-methylamino]dodecyl]indole-3-carbaldehyde |
NA |
177490 |
NA |
NA |
NA |
NA |
BindingDB |
| ACHE |
2-[(E)-2-[1-[[2-(trifluoromethyl)phenyl]methyl]-3,6-dihydro-2H-pyridin-4-yl]ethenyl]quinolin-8-ol;hydrochloride |
NA |
161000 |
NA |
NA |
NA |
NA |
BindingDB |
| ACHE |
Butyrylcholine |
NA |
229086.77 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ACHE |
2-(2-Chlorophenyl)-3-[3-(dimethylamino)propyl]-1,3-thiazolidin-4-one;hydrochloride |
NA|231000 |
134000|NA |
NA |
NA |
NA |
NA |
BindingDB |
| ACHE |
3-[3-(Dimethylamino)propyl]-2-pyridin-3-yl-1,3-thiazolidin-4-one;hydrochloride |
NA |
199000 |
NA |
NA |
NA |
NA |
BindingDB |
| ACHE |
3-[3-(Dimethylamino)propyl]-2-naphthalen-1-yl-1,3-thiazolidin-4-one;hydrochloride |
NA |
177000 |
NA |
NA |
NA |
NA |
BindingDB |
| ACHE |
(7R,13aS)-2,3,9-trimethoxy-7-methyl-6,8,13,13a-tetrahydro-5H-isoquinolino[2,1-b]isoquinolin-7-ium-4,10-diol;hydroxide |
NA |
131000 |
NA |
NA |
NA |
NA |
BindingDB |
| ACHE |
5-(bromomethyl)-N-pyridin-2-yl-4,5-dihydro-1,3-thiazol-2-amine;hydrobromide |
NA |
110000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ACHE |
Tacrine |
NA |
117000 |
NA |
NA |
NA |
NA |
BindingDB |
| ACHE |
N-(2-{[5-(furan-2-yl)-4-phenyl-4H-1,2,4-triazol-3-yl]sulfanyl}ethyl)benzenesulfonamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |