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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
ACHE 1-[4-(Pyridin-1-ium-1-yl)butyl]pyridin-1-ium dibromide NA 505000 NA NA NA NA TTD
ACHE 1,4-Bis(pyridinium)-butane dibromide NA 505000 NA NA NA NA BindingDB
ACHE 4-Chloro-N-[dichlorophosphinyl]benzamide NA 87000000 206000 NA NA NA BindingDB
ACHE 1,1'-(Oxydimethylene)bis(pyridinium chloride) NA 1770000 NA NA NA NA TTD
ACHE 1,3-Bis(pyridinium)-2-oxapropane dichloride NA 1770000 NA NA NA NA BindingDB
ACHE 1,1''-Bis(pyridinium)-1,3-phenyldimethylene dibromide NA 2360000 NA NA NA NA BindingDB
ACHE 1,1/'-(Oxydiethylene)dipyridinium dichloride NA 2010000 NA NA NA NA BindingDB
ACHE Butyrylthiocholine NA 125892.54 NA NA NA NA BindingDB|TTD
ACHE Alendronic Acid NA 27450000 NA NA NA NA BindingDB
ACHE Ladostigil NA 1000000 NA NA NA NA BindingDB
ACHE 2-[2-(2-Isoquinolin-2-ium-2-ylethoxy)ethyl]isoquinolin-2-ium;dibromide NA 1310000 NA NA NA NA TTD
ACHE N-(2-Morpholin-4-ylethyl)-6-phenyl-pyridazin-3-amine NA 1000000 NA NA NA NA BindingDB|TTD
ACHE Trimethyl(pent-4-enyl)azanium NA 1129795.91 NA NA NA NA BindingDB|TTD
ACHE (3-Acetylamino-phenyl)-trimethyl-ammonium; bromide NA 1000000 NA NA NA NA BindingDB|TTD
ACHE N,N-dimethyl-10H-phenothiazine-10-carboxamide 400000 NA NA NA NA NA BindingDB|TTD
ACHE N,N'-(3,3'-dimethylbiphenyl-4,4'-diyl)dibenzenesulfonamide NA 123110 NA NA NA NA BindingDB
ACHE 2-(4-Chloro-phenyl)-N-hydroxy-2-oxo-thioacetimidic acid 2-diethylamino-ethyl ester; hydrochloride NA 520000 NA NA NA NA BindingDB
ACHE Didecyldimonium Chloride NA NA NA NA 100262 NA PubChem
ACHE 10-O-Methylhostasine NA 113000 NA NA NA NA BindingDB|TTD
ACHE [3-(prop-2-ynylamino)-2,3-dihydro-1H-inden-4-yl] N-ethyl-N-methylcarbamate;hydrochloride NA 525000 NA NA NA NA TTD