GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
ACHE |
1-[4-(Pyridin-1-ium-1-yl)butyl]pyridin-1-ium dibromide |
NA |
505000 |
NA |
NA |
NA |
NA |
TTD |
ACHE |
1,4-Bis(pyridinium)-butane dibromide |
NA |
505000 |
NA |
NA |
NA |
NA |
BindingDB |
ACHE |
4-Chloro-N-[dichlorophosphinyl]benzamide |
NA |
87000000 |
206000 |
NA |
NA |
NA |
BindingDB |
ACHE |
1,1'-(Oxydimethylene)bis(pyridinium chloride) |
NA |
1770000 |
NA |
NA |
NA |
NA |
TTD |
ACHE |
1,3-Bis(pyridinium)-2-oxapropane dichloride |
NA |
1770000 |
NA |
NA |
NA |
NA |
BindingDB |
ACHE |
1,1''-Bis(pyridinium)-1,3-phenyldimethylene dibromide |
NA |
2360000 |
NA |
NA |
NA |
NA |
BindingDB |
ACHE |
1,1/'-(Oxydiethylene)dipyridinium dichloride |
NA |
2010000 |
NA |
NA |
NA |
NA |
BindingDB |
ACHE |
Butyrylthiocholine |
NA |
125892.54 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
ACHE |
Alendronic Acid |
NA |
27450000 |
NA |
NA |
NA |
NA |
BindingDB |
ACHE |
Ladostigil |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB |
ACHE |
2-[2-(2-Isoquinolin-2-ium-2-ylethoxy)ethyl]isoquinolin-2-ium;dibromide |
NA |
1310000 |
NA |
NA |
NA |
NA |
TTD |
ACHE |
N-(2-Morpholin-4-ylethyl)-6-phenyl-pyridazin-3-amine |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
ACHE |
Trimethyl(pent-4-enyl)azanium |
NA |
1129795.91 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
ACHE |
(3-Acetylamino-phenyl)-trimethyl-ammonium; bromide |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
ACHE |
N,N-dimethyl-10H-phenothiazine-10-carboxamide |
400000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
ACHE |
N,N'-(3,3'-dimethylbiphenyl-4,4'-diyl)dibenzenesulfonamide |
NA |
123110 |
NA |
NA |
NA |
NA |
BindingDB |
ACHE |
2-(4-Chloro-phenyl)-N-hydroxy-2-oxo-thioacetimidic acid 2-diethylamino-ethyl ester; hydrochloride |
NA |
520000 |
NA |
NA |
NA |
NA |
BindingDB |
ACHE |
Didecyldimonium Chloride |
NA |
NA |
NA |
NA |
100262 |
NA |
PubChem |
ACHE |
10-O-Methylhostasine |
NA |
113000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
ACHE |
[3-(prop-2-ynylamino)-2,3-dihydro-1H-inden-4-yl] N-ethyl-N-methylcarbamate;hydrochloride |
NA |
525000 |
NA |
NA |
NA |
NA |
TTD |