| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| SRC |
Ac-Cys-Ile-Tyr-Lys-Phe-Tyr-OH |
NA |
700000 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
Ac-Cys-Ile-Tyr-Lys-Tyr-Tyr-OH |
NA |
400000 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
3-(3,4-dichlorophenyl)-2-(4-hydroxyphenyl)-6,7-dihydro-5H-indazol-4-one |
NA |
150000 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
3-(3,4-Dichlorophenyl)-6,6-dimethyl-2-(4-nitrophenyl)-5,7-dihydroindazol-4-one |
NA |
150000 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
3-(4-Tert-butylphenyl)-6,6-dimethyl-2-(4-methylphenyl)-5,7-dihydroindazol-4-one |
NA |
150000 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
3-(3,4-dichlorophenyl)-2-(4-nitrophenyl)-6,7-dihydro-5H-indazol-4-one |
NA |
150000 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
3-(3,4-Dichlorophenyl)-2-(3-hydroxy-4-methoxyphenyl)-6,6-dimethyl-5,7-dihydroindazol-4-one |
NA |
150000 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
2-(4-Chlorophenyl)-3-cyclohexyl-6,6-dimethyl-[1,3]dioxino[4,5-c]pyrazol-4-one |
NA |
150000 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
3-(4-Tert-butylphenyl)-2-(3,4-dimethoxyphenyl)-6,6-dimethyl-5,7-dihydroindazol-4-one |
NA |
150000 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
3-(4-Tert-butylphenyl)-2-(4-chlorophenyl)-6,6-dimethyl-[1,3]dioxino[4,5-c]pyrazol-4-one |
NA |
150000 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
3-(3,4-dichlorophenyl)-2-(3-hydroxy-4-methoxyphenyl)-6,7-dihydro-5H-indazol-4-one |
NA |
150000 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
3-(4-Tert-butylphenyl)-2-(4-chlorophenyl)-6,6-dimethyl-5,7-dihydroindazol-4-one |
NA |
150000 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
3-(3,4-dichlorophenyl)-2-thiophen-2-yl-6,7-dihydro-5H-indazol-4-one |
NA |
150000 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
3-(3,4-dichlorophenyl)-2-(2-fluorophenyl)-6,7-dihydro-5H-indazol-4-one |
NA |
150000 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
3-(3-Chloro-4-methylphenyl)-2-(4-chlorophenyl)-6,6-dimethyl-5,7-dihydroindazol-4-one |
NA |
131800 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
3-Cyclohexyl-6,6-dimethyl-2-(4-nitrophenyl)-5,7-dihydroindazol-4-one |
NA |
150000 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
3-(3,4-dichlorophenyl)-2-(4-methylphenyl)-6,7-dihydro-5H-indazol-4-one |
NA |
150000 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
3-(3,4-dichlorophenyl)-2-(4-methoxyphenyl)-6,7-dihydro-5H-indazol-4-one |
NA |
150000 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
3-(3-chloro-4-methylphenyl)-6,6-dimethyl-2-(1H-pyrrol-2-yl)-5,7-dihydroindazol-4-one |
NA |
150000 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
3-(3,4-Dichlorophenyl)-6,6-dimethyl-2-thiophen-2-yl-5,7-dihydroindazol-4-one |
NA |
150000 |
NA |
NA |
NA |
NA |
TTD |