| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| SRC |
3-(3,4-Dichlorophenyl)-6,6-dimethyl-2-(4-methylphenyl)-5,7-dihydroindazol-4-one |
NA |
150000 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
3-(3,4-dichlorophenyl)-6,6-dimethyl-2-(1H-pyrrol-2-yl)-5,7-dihydroindazol-4-one |
NA |
150000 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
(2R,3S,4R,5S)-2-(hydroxymethyl)-5-(4-methoxyphenoxy)oxolane-3,4-diol |
NA |
483900 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
4-[(2S)-2-acetamido-2-{[(1S)-1-{3-[(4-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}ethyl]carbamoyl}ethyl]phenoxyphosphonic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
4-[(2S)-2-(1-phenylacetamido)-2-{[(1S)-1-(3-{[4-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)ethyl]carbamoyl}ethyl]phenoxyphosphonic acid |
NA |
123000 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
4-[(2S)-2-[1-(3,4-difluorophenyl)acetamido]-2-{[(1S)-1-(3-{[4-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)ethyl]carbamoyl}ethyl]phenoxyphosphonic acid |
NA |
130000 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
(2R,3S,4R,5R)-2-(hydroxymethyl)-5-naphthalen-1-yloxyoxolane-3,4-diol |
NA |
184700 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
6-(1,9-Diazaspiro[5.5]undecan-9-Yl)-9h-Purine |
NA |
150000 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
(2R,3S,4R,5R)-2-(hydroxymethyl)-5-naphthalen-2-yloxyoxolane-3,4-diol |
NA |
297300 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
(2R,3S,4R,5S)-2-(hydroxymethyl)-5-(4-phenylphenoxy)oxolane-3,4-diol |
NA |
125000 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
(2R,3S,4R,5R)-2-(hydroxymethyl)-5-(3-methylphenoxy)oxolane-3,4-diol |
NA |
451000 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
(2R,3S,4R,5S)-2-(hydroxymethyl)-5-naphthalen-2-yloxyoxolane-3,4-diol |
NA |
224800 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
(2R,3S,4R,5S)-2-(hydroxymethyl)-5-(4-methylphenoxy)oxolane-3,4-diol |
NA |
143400 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
Src SH2 inhibitor, 1h |
NA |
335000 |
NA |
NA |
NA |
NA |
BindingDB |
| SRC |
N-hydroxy-6-(5-phenyltriazol-1-yl)hexanamide |
12500000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| SRC |
AC-Dopa-eee |
NA |
160000 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
cyclo[Lys-Phe-Lys-Phe-Lys-Phe-Lys-Phe] |
NA |
1567600 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
Phenylmalonic acid |
NA |
2500000|200000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SRC |
2-Naphthyl dihydrogen phosphate |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
p-tert-Butylphenyl dihydrogen phosphate |
NA |
4000000 |
NA |
NA |
NA |
NA |
TTD |