| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| SRC |
4-[(2S)-2-{[(1S)-3-carbamoyl-1-[3-(naphthalen-2-ylmethyl)-1,2,4-oxadiazol-5-yl]propyl]carbamoyl}-2-acetamidoethyl]phenoxyphosphonic acid |
NA |
274000 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
4-[(2S)-2-acetamido-2-{[(1S)-2-hydroxy-1-(3-{[4-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)ethyl]carbamoyl}ethyl]phenoxyphosphonic acid |
NA |
282000 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
4-[(2S)-2-{[(1S)-2-hydroxy-1-(3-{[4-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)ethyl]carbamoyl}-2-(1-phenylacetamido)ethyl]phenoxyphosphonic acid |
NA |
161000 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
1-(4-Chlorophenyl)-2-(4-(thiophen-3-yl)-1H-1,2,3-triazol-1-yl)ethanone |
NA |
150000 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
N-ethyl-2-(4-phenyl-1H-1,2,3-triazol-1-yl)acetamide |
NA |
150000 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
1-(4-phenyl-1H-1,2,3-triazol-1-yl)propan-2-one |
NA |
150000 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
1-(4-p-tolyl-1H-1,2,3-triazol-1-yl)propan-2-one |
NA |
150000 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
3-(2-(4-p-Tolyl-1H-1,2,3-triazol-1-yl)acetyl)-2H-chromen-2-one |
NA |
150000 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
1-(4-chlorophenyl)-2-(4-p-tolyl-1H-1,2,3-triazol-1-yl)ethanone |
NA |
108700 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
2-(4-phenyl-1H-1,2,3-triazol-1-yl)cyclopentanone |
NA |
105500 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
N-((5-Methoxy-1H-indol-3-yl)(p-tolyl)methyl)-N-methylbenzenamine |
NA |
150000 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
N-((5-Bromo-1H-indol-3-yl)(p-tolyl)methyl)-N-methylbenzenamine |
NA |
150000 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
N-((5-bromo-1H-indol-3-yl)(4-methoxyphenyl)methyl)-N-methylaniline |
NA |
106000 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
N-((1H-Indol-3-yl)(3-methoxyphenyl)methyl)-N-methylbenzenamine |
NA |
150000 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
N-((1H-Indol-3-yl)(4-methoxyphenyl)methyl)-N-methylbenzenamine |
NA |
150000 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
N-((1H-Indol-3-yl)(4-hydroxy phenyl)methyl)-N-methylbenzenamine |
NA |
150000 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
N-((1H-Indol-3-yl)(2,4-dimethoxyphenyl)methyl)-N-methylbenzenamine |
NA |
150000 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
N-Methyl-N-((1-methyl-1H-indol-3-yl)(phenyl)methyl)benzenamine |
NA |
150000 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
N-((1H-Indol-3-yl)(p-tolyl)methyl)-N-methylbenzenamine |
NA |
150000 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
N-((4-Hydroxy-3-bromophenyl)(1H-indol-3-yl)methyl)-N-methylbenzenamine |
NA |
150000 |
NA |
NA |
NA |
NA |
TTD |