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drugs and pathways
negative DTIs
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Drugs And Genes
Negative Drug Target Genes
Gene
Drug
GENE_SYMBOL
DRUG_NAME
Ki (nM)
IC50 (nM)
Kd (nM)
EC50 (nM)
Potency (nM)
AC50 (nM)
Datasource
SRC
Tpl2-IN-I
NA
400000000
NA
NA
NA
NA
TTD
SRC
[(3,4,5-Trimethoxyphenyl)amino]carbonylphosphonic acid
NA
2100000
NA
NA
NA
NA
TTD
SRC
{[2-(Trifluoromethoxy)phenyl]amino}carbonylphosphonic acid
NA
4000000
NA
NA
NA
NA
TTD
SRC
[(4-Butoxyphenyl)amino]carbonylphosphonic acid
NA
3900000
NA
NA
NA
NA
TTD
SRC
{[4-(Ethoxycarbonyl)phenyl]amino}carbonylphosphonic acid
NA
3600000
NA
NA
NA
NA
TTD
SRC
Phosphoric acid 2-formyl-phenyl ester methyl ester
NA
3300000
NA
NA
NA
NA
TTD
SRC
Phosphoric acid 4-(trifluoromethylthio)phenyl ester
NA
1200000
NA
NA
NA
NA
TTD
SRC
Phosphoric acid mono-(8-hydroxy-3,4-dihydro-2H-quinolin-1-yl) ester
NA
300000
NA
NA
NA
NA
TTD
SRC
Phosphoric acid mono-(2-acetyl-naphthalen-1-yl) ester
NA
3500000
NA
NA
NA
NA
TTD
SRC
3-Phosphonooxy-naphthalene-2-carboxylic acid methyl ester
NA
3200000
NA
NA
NA
NA
TTD
SRC
3-Phosphonooxy-benzoic acid methyl ester
NA
4000000
NA
NA
NA
NA
TTD
SRC
Phosphoric acid mono-(3-formyl-phenyl) ester
NA
600000
NA
NA
NA
NA
TTD
SRC
Ac-YEEIE
NA
200000
NA
NA
NA
NA
TTD
SRC
RU79072
NA
3600000
NA
NA
NA
NA
BindingDB|TTD
SRC
Iso24
NA
4400000
NA
NA
NA
NA
BindingDB|TTD
SRC
RU78783
NA
3900000
NA
NA
NA
NA
BindingDB|TTD
SRC
1-(4-chlorophenyl)-2-(4-phenyl-1H-1,2,3-triazol-1-yl)ethanone
NA
139000
NA
NA
NA
NA
TTD
SRC
1-[2-(Furan-2-yl)pyrrolidin-1-yl]prop-2-en-1-one
160000
NA
NA
NA
NA
NA
ChEMBL|TTD
SRC
Pas219
NA
2300000
NA
NA
NA
NA
BindingDB|TTD
SRC
RU78262
NA
300000
NA
NA
NA
NA
BindingDB
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