| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| SRC |
[4-[(2S)-2-acetamido-3-[[(1S)-4-amino-1-(3-butyl-1,2,4-oxadiazol-5-yl)-4-oxobutyl]amino]-3-oxopropyl]phenyl] dihydrogen phosphate |
NA |
384000 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
[4-[(2S)-2-acetamido-3-[[(1S)-4-amino-1-[3-(3-methylbutyl)-1,2,4-oxadiazol-5-yl]-4-oxobutyl]amino]-3-oxopropyl]phenyl] dihydrogen phosphate |
NA |
320000 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
[4-[(2S)-2-acetamido-3-[[(1S)-1-[3-(3-methylbutyl)-1,2,4-oxadiazol-5-yl]propyl]amino]-3-oxopropyl]phenyl] dihydrogen phosphate |
NA |
111000 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
Phosphoric acid mono-(4-formyl-2,6-dimethyl-phenyl) ester |
NA |
5000000 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
[5-[[(1S)-1-[3-[(3,4-dichlorophenyl)methyl]-1,2,4-oxadiazol-5-yl]ethyl]carbamoylamino]naphthalen-2-yl] dihydrogen phosphate |
NA |
198000 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
Ac-Tyr(PO3H2)-Asn-Glu-Leu-NH2 |
NA |
237000 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
[4-[(2S)-2-acetamido-3-[[(1S)-4-amino-4-oxo-1-[3-[(4,6,6-trimethylcyclohexa-2,4-dien-1-yl)methyl]-1,2,4-oxadiazol-5-yl]butyl]amino]-3-oxopropyl]phenyl] dihydrogen phosphate |
NA |
312000 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
Ac-Tyr(PO3H2)-Asp-Val-Leu-NH2 |
NA |
261000 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
Ac-Lys(1)-D-Tyr(PO3H2)-Val-D-Asn-Cha-D-Pro-(1) |
NA |
150000 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
Ac-Lys(1)-D-Tyr(PO3H2)-Cha-D-Asn-Val-D-Pro-(1) |
NA |
150000 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
Ac-Lys(1)-D-Tyr(PO3H2)-Leu-D-Asn-Val-D-Pro-(1) |
NA |
150000 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
Ac-Lys(1)-D-Tyr(PO3H2)-Val-D-Asn-Val-D-Pro-(1) |
NA |
150000 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
5-{[(S)-1-(4-Methoxy-benzylcarbamoyl)-3-methyl-butylcarbamoyl]-methoxy}-isophthalic acid |
NA |
864000 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
4-{[(S)-1-(3-Methoxy-benzylcarbamoyl)-2-methyl-propylcarbamoyl]-methoxy}-pyridine-2,6-dicarboxylic acid dimethyl ester |
NA |
713000 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
4-({(S)-1-[(Benzo[1,3]dioxol-5-ylmethyl)-carbamoyl]-2-phenyl-ethylcarbamoyl}-methoxy)-pyridine-2,6-dicarboxylic acid dimethyl ester |
NA |
396000 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
4-[({(S)-[(Benzo[1,3]dioxol-5-ylmethyl)-carbamoyl]-phenyl-methyl}-carbamoyl)-methoxy]-pyridine-2,6-dicarboxylic acid dimethyl ester |
NA |
714000 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
4-{[(S)-1-(3-Methoxy-benzylcarbamoyl)-2-phenyl-ethylcarbamoyl]-methoxy}-pyridine-2,6-dicarboxylic acid dimethyl ester |
NA |
663000 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
Ac-Cys-Tyr-Lys-Tyr(4-PO3H2)-Tyr |
NA |
700000 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
Ac-Cys-Ile-Tyr-Lys-Tyr(4-PO3H2)-Tyr |
NA |
700000 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
N-Methyl-N,5-diphenylimidazo[1,5-A]pyrazin-8-amine |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |