GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
SRC |
3,5-Dihydroxy-N-(3-hydroxyphenyl)naphthalene-2-carboxamide |
NA |
150000 |
NA |
NA |
NA |
NA |
TTD |
SRC |
Naphthyl phosphate |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
SRC |
Phosphoric acid mono-(2,6-dimethyl-phenyl) ester |
NA |
10000000 |
NA |
NA |
NA |
NA |
TTD |
SRC |
[Hydroxy-(6-nitro-1,3-benzodioxol-5-yl)methyl]phosphonic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
SRC |
N-(4-Methyl-3-(2-(6-(methylamino)-9H-purin-9-yl)ethyl)phenyl)-3-(trifluoromethyl)-benzamide |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
SRC |
Citric Acid |
NA |
40000000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
SRC |
(4-Hydroxy-phenyl)-sulfo-acetic acid |
NA |
190000 |
NA |
NA |
NA |
NA |
TTD |
SRC |
Fosfosal |
NA |
2000000 |
NA |
NA |
NA |
NA |
TTD |
SRC |
4-Nitrophenyl Phosphate |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
SRC |
alpha-Sulfophenylacetic acid |
NA |
3200000 |
NA |
NA |
NA |
NA |
BindingDB |
SRC |
8-chloro-4-(3-chloro-4-fluorophenylamino)-6-((1-(1-cyclobutylpiperidin-4-yl)-1H-1,2,3-triazol-4-yl)methylamino)quinoline-3-carbonitrile |
NA |
110000 |
NA |
NA |
NA |
NA |
TTD |
SRC |
N-((4-Chlorophenyl)(1H-indol-3-yl)methyl)-N-methylbenzenamine |
NA |
150000 |
NA |
NA |
NA |
NA |
TTD |
SRC |
(2R,3S,4R,5S)-2-(hydroxymethyl)-5-(4-hydroxyphenoxy)oxolane-3,4-diol |
NA |
272100 |
NA |
NA |
NA |
NA |
TTD |
SRC |
N-[3-[(E)-2-[6-[3-(dimethylamino)propylamino]purin-9-yl]ethenyl]-4-methylphenyl]-3-(trifluoromethyl)benzamide |
NA |
159000 |
NA |
NA |
NA |
NA |
TTD |
SRC |
(E)-N-(4-Methyl-3-(2-(6-(pyridine-2-yl-amino)-9H-purin-9-yl)vinyl)phenyl)-3-(trifluoromethyl)-benzamide |
NA |
201000 |
NA |
NA |
NA |
NA |
TTD |
SRC |
N-(5-tert-butyl-1,3-thiazol-2-yl)-3-[(E)-2-[6-(cyclopropylamino)purin-9-yl]ethenyl]-4-methylbenzamide |
NA |
310000 |
NA |
NA |
NA |
NA |
TTD |
SRC |
(E)-1-(3-(2-(6-(Cyclopropylamino)-9H-purin-9-yl)vinyl)-4-methylphenyl)-3-(3-(trifluoromethyl)phenyl)urea |
NA |
517000 |
NA |
NA |
NA |
NA |
TTD |
SRC |
7,8-Dimethoxy-3-(2-morpholin-4-yl-ethyl)-5,10-dihydro-3H-pyrimido[4,5-b]quinolin-4-one |
NA |
105000 |
NA |
NA |
NA |
NA |
TTD |
SRC |
Phosphoric acid 2-formyl-phenyl ester isopropyl ester |
NA |
2100000 |
NA |
NA |
NA |
NA |
TTD |
SRC |
Phosphoric acid mono-(2,6-diformyl-phenyl) ester |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |