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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
SQLE 5,9,14,18-Tetramethyl-docosa-5,9,13,17-tetraene-1,21-diyne NA 400000 NA NA NA NA TTD
SQLE 6,10,15,19,23-Pentamethyl-tetracosa-6,10,14,18,22-pentaen-1-yn-3-ol NA|950000 400000|NA NA NA NA NA BindingDB|TTD
SQLE 6,10,15,19-Tetramethyl-tetracosa-6,10,14,18-tetraene-1,23-diyne-3,22-diol 1000000|NA NA|400000 NA NA NA NA BindingDB|TTD
SQLE (4,8,13,17,21-Pentamethyl-docosa-4,8,12,16,20-pentaenylidene)-cyclopropane NA 400000 NA NA NA NA TTD
SQLE (1,5,9,14,18,22-Hexamethyl-tricosa-1,5,9,13,17,21-hexaenyl)-cyclopropane NA 400000 NA NA NA NA TTD
SQLE 4,8,12,17,21,25-Hexamethyl-hexacosa-4,8,12,16,20,24-hexaen-1-ol NA 400000 NA NA NA NA TTD
SQLE (1E,5E,9E,13E,17E)-5,9,14,18,22-Pentamethyl-1-nitro-tricosa-1,5,9,13,17,21-hexaene NA 400000 NA NA NA NA TTD
SQLE (9E,13E,21E)-5,9,14,18,22-Pentamethyl-1-nitro-tricosa-5,9,13,17,21-pentaen-1-ol NA 270000 NA NA NA NA BindingDB|TTD
SQLE [4-(Chloromethyl)phenyl]-[4-[ethyl-[[3-[(4-thiophen-2-ylthiophen-2-yl)methoxy]phenyl]methyl]amino]phenyl]methanone NA 500000 NA NA NA NA BindingDB|TTD
SQLE [3-[[3-[[[(E)-6,6-dimethylhept-2-en-4-ynyl]-ethylamino]methyl]phenoxy]methyl]-5-[3-(trifluoromethyl)diazirin-3-yl]phenyl]methanol NA 500000 NA NA NA NA BindingDB|TTD
SQLE 3-[Ethyl-[[3-[(4-thiophen-2-ylthiophen-2-yl)methoxy]phenyl]methyl]amino]-5-[3-(trifluoromethyl)diazirin-3-yl]phenol NA 500000 NA NA NA NA BindingDB|TTD
SQLE 2-[Ethyl-[[3-[(4-thiophen-2-ylthiophen-2-yl)methoxy]phenyl]methyl]amino]-4-[3-(trifluoromethyl)diazirin-3-yl]phenol NA 500000 NA NA NA NA BindingDB|TTD
SQLE (2Z,10E,14E)-6,11,15,19-tetramethyl-2-(4-methylpent-3-enyl)icosa-2,6,10,14,18-pentaen-1-amine NA 109000 NA NA NA NA BindingDB
SQLE 4,8,12-Tetradecatrien-1-ol, 5,9,13-trimethyl- NA 400000 NA NA NA NA TTD
SRC 3-[[4-(3-Pyridinyl)-2-pyrimidinyl]amino]benzoic acid NA 126000 NA NA NA NA TTD
SRC Phosphoric Acid NA 40000000 NA NA NA NA PubChem|TTD
SRC [4-[(2S)-2-acetamido-3-[[3-(cyclohexylmethyl)phenyl]methylamino]-3-oxopropyl]phenyl] dihydrogen phosphate NA 769000 NA NA NA NA TTD
SRC (2-Formyl-4-methyl-phenyl)-acetic acid NA 385000 NA NA NA NA TTD
SRC Ac-Cys-Ile-Tyr-Lys-Phe(4-NHMes)-Tyr-OH NA 700000 NA NA NA NA TTD
SRC (E)-N-(4-((3-chloro-4-fluorophenyl)amino)-7-methoxyquinazolin-6-yl)-4-(piperidin-1-yl)but-2-enamide NA 110000 NA NA NA NA PubChem