GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
SQLE |
5,9,14,18-Tetramethyl-docosa-5,9,13,17-tetraene-1,21-diyne |
NA |
400000 |
NA |
NA |
NA |
NA |
TTD |
SQLE |
6,10,15,19,23-Pentamethyl-tetracosa-6,10,14,18,22-pentaen-1-yn-3-ol |
NA|950000 |
400000|NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SQLE |
6,10,15,19-Tetramethyl-tetracosa-6,10,14,18-tetraene-1,23-diyne-3,22-diol |
1000000|NA |
NA|400000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SQLE |
(4,8,13,17,21-Pentamethyl-docosa-4,8,12,16,20-pentaenylidene)-cyclopropane |
NA |
400000 |
NA |
NA |
NA |
NA |
TTD |
SQLE |
(1,5,9,14,18,22-Hexamethyl-tricosa-1,5,9,13,17,21-hexaenyl)-cyclopropane |
NA |
400000 |
NA |
NA |
NA |
NA |
TTD |
SQLE |
4,8,12,17,21,25-Hexamethyl-hexacosa-4,8,12,16,20,24-hexaen-1-ol |
NA |
400000 |
NA |
NA |
NA |
NA |
TTD |
SQLE |
(1E,5E,9E,13E,17E)-5,9,14,18,22-Pentamethyl-1-nitro-tricosa-1,5,9,13,17,21-hexaene |
NA |
400000 |
NA |
NA |
NA |
NA |
TTD |
SQLE |
(9E,13E,21E)-5,9,14,18,22-Pentamethyl-1-nitro-tricosa-5,9,13,17,21-pentaen-1-ol |
NA |
270000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SQLE |
[4-(Chloromethyl)phenyl]-[4-[ethyl-[[3-[(4-thiophen-2-ylthiophen-2-yl)methoxy]phenyl]methyl]amino]phenyl]methanone |
NA |
500000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SQLE |
[3-[[3-[[[(E)-6,6-dimethylhept-2-en-4-ynyl]-ethylamino]methyl]phenoxy]methyl]-5-[3-(trifluoromethyl)diazirin-3-yl]phenyl]methanol |
NA |
500000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SQLE |
3-[Ethyl-[[3-[(4-thiophen-2-ylthiophen-2-yl)methoxy]phenyl]methyl]amino]-5-[3-(trifluoromethyl)diazirin-3-yl]phenol |
NA |
500000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SQLE |
2-[Ethyl-[[3-[(4-thiophen-2-ylthiophen-2-yl)methoxy]phenyl]methyl]amino]-4-[3-(trifluoromethyl)diazirin-3-yl]phenol |
NA |
500000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SQLE |
(2Z,10E,14E)-6,11,15,19-tetramethyl-2-(4-methylpent-3-enyl)icosa-2,6,10,14,18-pentaen-1-amine |
NA |
109000 |
NA |
NA |
NA |
NA |
BindingDB |
SQLE |
4,8,12-Tetradecatrien-1-ol, 5,9,13-trimethyl- |
NA |
400000 |
NA |
NA |
NA |
NA |
TTD |
SRC |
3-[[4-(3-Pyridinyl)-2-pyrimidinyl]amino]benzoic acid |
NA |
126000 |
NA |
NA |
NA |
NA |
TTD |
SRC |
Phosphoric Acid |
NA |
40000000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
SRC |
[4-[(2S)-2-acetamido-3-[[3-(cyclohexylmethyl)phenyl]methylamino]-3-oxopropyl]phenyl] dihydrogen phosphate |
NA |
769000 |
NA |
NA |
NA |
NA |
TTD |
SRC |
(2-Formyl-4-methyl-phenyl)-acetic acid |
NA |
385000 |
NA |
NA |
NA |
NA |
TTD |
SRC |
Ac-Cys-Ile-Tyr-Lys-Phe(4-NHMes)-Tyr-OH |
NA |
700000 |
NA |
NA |
NA |
NA |
TTD |
SRC |
(E)-N-(4-((3-chloro-4-fluorophenyl)amino)-7-methoxyquinazolin-6-yl)-4-(piperidin-1-yl)but-2-enamide |
NA |
110000 |
NA |
NA |
NA |
NA |
PubChem |