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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
SRC Cyclo[Ac-Cys-Ile-Tyr-Lys-Phe]-Tyr NA 400000 NA NA NA NA TTD
SRC Ac-Cys-Ile-Phe(4-NH2)-Lys-Tyr-Tyr-OH NA 760000 NA NA NA NA TTD
SRC Ac-Cys-Ile-Tyr-Lys-Phe(4-guanidino)-Tyr-OH NA 700000 NA NA NA NA TTD
SRC (2S)-2-[[(2S)-2-[[(3S,6S,9R,20S)-6-[(2S)-butan-2-yl]-3-[(4-hydroxyphenyl)methyl]-2,5,8,11,14-pentaoxo-9-(sulfanylmethyl)-1,4,7,10,15-pentazacycloicosane-20-carbonyl]amino]-3-(4-nitrophenyl)propanoyl]amino]-3-(4-hydroxyphenyl)propanoic acid NA 134000 NA NA NA NA TTD
SRC (2S)-2-[[(12S,15S)-12-[[(2S)-2-[[(2S,3S)-2-[[(2R)-2-acetamido-3-sulfanylpropanoyl]amino]-3-methylpentanoyl]amino]-3-(4-hydroxyphenyl)propanoyl]amino]-3,6,13-trioxo-2,7,14-triazabicyclo[15.2.2]henicosa-1(19),17,20-triene-15-carbonyl]amino]-3-(4-hydroxyphenyl)propanoic acid NA 400000 NA NA NA NA TTD
SRC Ac-Cys-Ile-Tyr-Lys-Tyr-Phe(4-NH2)-OH NA 700000 NA NA NA NA TTD
SRC {[4-(Benzyloxy)phenyl]amino}carbonylphosphonic acid NA 800000 NA NA NA NA TTD
SRC 4-Aminophenyl phosphate NA 600000 NA NA NA NA TTD
SRC Phosphoric acid mono-m-tolyl ester NA 4000000 NA NA NA NA TTD
SRC Phosphoric acid mono-p-tolyl ester NA 2000000 NA NA NA NA TTD
SRC p-Methoxyphenyl dihydrogen phosphate NA 4000000 NA NA NA NA TTD
SRC 4-Phosphonooxy-benzoic acid methyl ester NA 4000000 NA NA NA NA TTD
SRC Phenylphosphate NA 3500000 NA NA NA NA BindingDB|TTD
SRC [4-[3-[[(1S)-1-[3-[(3,4-dichlorophenyl)methyl]-1,2,4-oxadiazol-5-yl]ethyl]amino]-3-oxopropyl]phenyl] dihydrogen phosphate NA 459000 NA NA NA NA TTD
SRC [4-[(2S)-2-(tert-butylsulfonylmethyl)-3-oxo-3-[[(1S)-1-[3-[[4-(trifluoromethyl)phenyl]methyl]-1,2,4-oxadiazol-5-yl]ethyl]amino]propyl]phenyl] dihydrogen phosphate NA 205000 NA NA NA NA TTD
SRC 3H,4H,9H-pyrimido[4,5-b]indol-4-one NA 293000 NA NA NA NA TTD
SRC 10-Ethyl-5,10-dihydro-3H-pyrimido[4,5-b]quinolin-4-one NA 550000 NA NA NA NA TTD
SRC 6-(Phenylamino)pyrimidin-4-ol NA 1550000 NA NA NA NA TTD
SRC Chlorophenol phosphate NA 3500000 NA NA NA NA TTD
SRC alpha-naphthyl beta-D-ribofuranoside NA 1370700 NA NA NA NA TTD