GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
SRC |
Cyclo[Ac-Cys-Ile-Tyr-Lys-Phe]-Tyr |
NA |
400000 |
NA |
NA |
NA |
NA |
TTD |
SRC |
Ac-Cys-Ile-Phe(4-NH2)-Lys-Tyr-Tyr-OH |
NA |
760000 |
NA |
NA |
NA |
NA |
TTD |
SRC |
Ac-Cys-Ile-Tyr-Lys-Phe(4-guanidino)-Tyr-OH |
NA |
700000 |
NA |
NA |
NA |
NA |
TTD |
SRC |
(2S)-2-[[(2S)-2-[[(3S,6S,9R,20S)-6-[(2S)-butan-2-yl]-3-[(4-hydroxyphenyl)methyl]-2,5,8,11,14-pentaoxo-9-(sulfanylmethyl)-1,4,7,10,15-pentazacycloicosane-20-carbonyl]amino]-3-(4-nitrophenyl)propanoyl]amino]-3-(4-hydroxyphenyl)propanoic acid |
NA |
134000 |
NA |
NA |
NA |
NA |
TTD |
SRC |
(2S)-2-[[(12S,15S)-12-[[(2S)-2-[[(2S,3S)-2-[[(2R)-2-acetamido-3-sulfanylpropanoyl]amino]-3-methylpentanoyl]amino]-3-(4-hydroxyphenyl)propanoyl]amino]-3,6,13-trioxo-2,7,14-triazabicyclo[15.2.2]henicosa-1(19),17,20-triene-15-carbonyl]amino]-3-(4-hydroxyphenyl)propanoic acid |
NA |
400000 |
NA |
NA |
NA |
NA |
TTD |
SRC |
Ac-Cys-Ile-Tyr-Lys-Tyr-Phe(4-NH2)-OH |
NA |
700000 |
NA |
NA |
NA |
NA |
TTD |
SRC |
{[4-(Benzyloxy)phenyl]amino}carbonylphosphonic acid |
NA |
800000 |
NA |
NA |
NA |
NA |
TTD |
SRC |
4-Aminophenyl phosphate |
NA |
600000 |
NA |
NA |
NA |
NA |
TTD |
SRC |
Phosphoric acid mono-m-tolyl ester |
NA |
4000000 |
NA |
NA |
NA |
NA |
TTD |
SRC |
Phosphoric acid mono-p-tolyl ester |
NA |
2000000 |
NA |
NA |
NA |
NA |
TTD |
SRC |
p-Methoxyphenyl dihydrogen phosphate |
NA |
4000000 |
NA |
NA |
NA |
NA |
TTD |
SRC |
4-Phosphonooxy-benzoic acid methyl ester |
NA |
4000000 |
NA |
NA |
NA |
NA |
TTD |
SRC |
Phenylphosphate |
NA |
3500000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SRC |
[4-[3-[[(1S)-1-[3-[(3,4-dichlorophenyl)methyl]-1,2,4-oxadiazol-5-yl]ethyl]amino]-3-oxopropyl]phenyl] dihydrogen phosphate |
NA |
459000 |
NA |
NA |
NA |
NA |
TTD |
SRC |
[4-[(2S)-2-(tert-butylsulfonylmethyl)-3-oxo-3-[[(1S)-1-[3-[[4-(trifluoromethyl)phenyl]methyl]-1,2,4-oxadiazol-5-yl]ethyl]amino]propyl]phenyl] dihydrogen phosphate |
NA |
205000 |
NA |
NA |
NA |
NA |
TTD |
SRC |
3H,4H,9H-pyrimido[4,5-b]indol-4-one |
NA |
293000 |
NA |
NA |
NA |
NA |
TTD |
SRC |
10-Ethyl-5,10-dihydro-3H-pyrimido[4,5-b]quinolin-4-one |
NA |
550000 |
NA |
NA |
NA |
NA |
TTD |
SRC |
6-(Phenylamino)pyrimidin-4-ol |
NA |
1550000 |
NA |
NA |
NA |
NA |
TTD |
SRC |
Chlorophenol phosphate |
NA |
3500000 |
NA |
NA |
NA |
NA |
TTD |
SRC |
alpha-naphthyl beta-D-ribofuranoside |
NA |
1370700 |
NA |
NA |
NA |
NA |
TTD |