| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| SRC |
RU78299 |
NA |
500000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SRC |
RU78300 |
NA |
900000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SRC |
RU79073 |
NA |
300000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SRC |
Pasbn |
NA |
1200000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SRC |
Phenanthridinone deriv. 5j |
NA |
197000 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
4-[(2S)-2-{[(1S)-3-carbamoyl-1-{3-[(4-methylphenyl)methyl]-1,2,4-oxadiazol-5-yl}propyl]carbamoyl}-2-acetamidoethyl]phenoxyphosphonic acid |
NA |
292000 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
4-[(2S)-2-{[(1S)-3-carbamoyl-1-{3-[(4-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}propyl]carbamoyl}-2-acetamidoethyl]phenoxyphosphonic acid |
NA |
205000 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
4-[(2S)-2-{[(1S)-3-carbamoyl-1-{3-[(3-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}propyl]carbamoyl}-2-acetamidoethyl]phenoxyphosphonic acid |
NA |
259000 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
4-[(2S)-2-{[(1S)-3-carbamoyl-1-{3-[(2,4-dichlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}propyl]carbamoyl}-2-acetamidoethyl]phenoxyphosphonic acid |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
4-[(2S)-2-{[(1S)-3-carbamoyl-1-[3-(naphthalen-1-ylmethyl)-1,2,4-oxadiazol-5-yl]propyl]carbamoyl}-2-acetamidoethyl]phenoxyphosphonic acid |
NA |
135000 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
4-[(2S)-2-{[(1S)-3-carbamoyl-1-[3-(2-phenylethyl)-1,2,4-oxadiazol-5-yl]propyl]carbamoyl}-2-acetamidoethyl]phenoxyphosphonic acid |
NA |
156000 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
4-[(2S)-2-acetamido-2-{[(1S)-1-(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)ethyl]carbamoyl}ethyl]phenoxyphosphonic acid |
NA |
115000 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
4-[(2S)-2-acetamido-2-{[2-(3-{[4-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)propan-2-yl]carbamoyl}ethyl]phenoxyphosphonic acid |
NA |
489000 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
4-[(2S)-2-acetamido-2-{[(3-{[4-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]carbamoyl}ethyl]phenoxyphosphonic acid |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
4-[(2S)-2-acetamido-2-{[2-(3-{[4-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)ethyl]carbamoyl}ethyl]phenoxyphosphonic acid |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
4-[(2S)-2-{[(1S)-2-carbamoyl-1-(3-{[4-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)ethyl]carbamoyl}-2-acetamidoethyl]phenoxyphosphonic acid |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
4-[(2S)-2-{[(1S)-1-{3-[(4-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}-2-hydroxyethyl]carbamoyl}-2-acetamidoethyl]phenoxyphosphonic acid |
NA |
149000 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
4-[(2S)-2-acetamido-2-{[(1S)-1-{3-[(4-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}-2-hydroxyethyl]carbamoyl}ethyl]phenoxyphosphonic acid |
NA |
132000 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
4-[(2S)-2-[1-(thiophen-2-yl)acetamido]-2-{[(1S)-1-(3-{[4-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)ethyl]carbamoyl}ethyl]phenoxyphosphonic acid |
NA |
143000 |
NA |
NA |
NA |
NA |
TTD |
| SRC |
4-[(2S)-2-{[(1S)-3-carbamoyl-1-{3-[(3,4-dichlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}propyl]carbamoyl}-2-acetamidoethyl]phenoxyphosphonic acid |
NA |
206000 |
NA |
NA |
NA |
NA |
TTD |