GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
SRPK1 |
Kinase inhibitor, A1 |
NA |
114000 |
NA |
NA |
NA |
NA |
BindingDB |
SRR |
(2S)-2-[(4-nitrophenyl)sulfonylamino]butanoic acid |
1500000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SRR |
(S)-2-((S)-3-(1H-imidazol-4-yl)-2-(3-phenylpropanamido)propanamido)-4-phenylbutanamide |
320000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SRR |
3-(Carboxymethyl)quinuclidine-3-carboxylic acid |
10000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
SRR |
(2S,3R)-2-((S)-3-(1H-imidazol-4-yl)-2-(3-phenylpropanamido)propanamido)-3-methylpentanamide |
610000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SRR |
Thiophen-2-ylsulfonylmethylcarbamic acid |
1500000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SRR |
2-[3-[3-(2-Hydroxyethylsulfanyl)-5-nitrophenyl]-2-oxopropoxy]acetic acid |
4500000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SRR |
3-Hydroxycoumarin |
NA |
10000000 |
NA |
NA |
NA |
NA |
TTD |
SRR |
[2-(4-Acetamidoanilino)-2-oxoethyl] 3-(2-methoxyphenyl)sulfanylpropanoate |
NA |
836000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SRR |
Tricarballylic Acid |
1300000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SRR |
4,5,6,7-Tetrahydro-1-benzothiophene-2-carboxylic acid |
NA |
5015000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SRR |
4-Ethyl-5-propylthiophene-2-carboxylic acid |
NA |
10000000 |
NA |
NA |
NA |
NA |
TTD |
SRR |
Benzoic Acid |
NA |
10000000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
SRR |
4-Ethyl-5-methylthiophene-2-carboxylic acid |
NA |
5723000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SRR |
N-[(1,3-dimethyl-2,4,6-trioxotetrahydro-5(2H)-pyrimidinylidene)methyl]aspartic acid |
1700000 |
NA |
NA |
NA |
NA |
NA |
TTD |
SRR |
2-Phenyl-1,3,4-oxadiazol-2-IN-5-one |
NA |
10000000 |
NA |
NA |
NA |
NA |
TTD |
SRR |
5-Methyl-4-propylthiophene-2-carboxylic acid |
NA |
5159000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SRR |
meso-Tartaric acid |
NA |
2820000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SRR |
|
1700000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
SRR |
Crotonic acid |
NA |
10000000 |
NA |
NA |
NA |
NA |
TTD |