| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| SRR |
3'-Hydroxycinnamic acid |
NA |
8386000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| SRR |
3-Thiophenecarboxylic acid |
NA |
8213000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SRR |
Glycine |
366000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| SRR |
2-[[2-(4-chlorophenoxy)acetyl]amino]-N-(2,3,4-trifluorophenyl)acetamide |
NA |
140000|1210000|1603000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SRR |
4H,5H,6H-cyclopenta(b)thiophene-2-carboxylic acid |
NA |
5282000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SRR |
5-(2-methylphenyl)-3H-1,3,4-oxadiazol-2-one |
NA |
5000000 |
NA |
NA |
NA |
NA |
TTD |
| SRR |
Malonic acid |
NA |
1310000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
| SRR |
2-[[2-(4-bromophenoxy)acetyl]amino]-N-(2,6-difluorophenyl)acetamide |
NA |
630000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SRR |
N-(4-bromophenyl)-2-[[2-(4-fluorophenoxy)acetyl]amino]acetamide |
NA |
520000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SSTR1 |
1-(4-aminobutyl)-8-benzyl-12-[(2R)-2-hydroxypropyl]-4-[2-(1H-indol-3-yl)ethyl]-1,4,8,12-tetrazacyclopentadecane-2,5,9,13-tetrone |
153000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| SSTR1 |
1-(4-aminobutyl)-9-benzyl-13-[(2R)-2-hydroxypropyl]-5-[2-(1H-indol-3-yl)ethyl]-1,5,9,13-tetrazacyclohexadecane-2,6,10,14-tetrone |
102000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| SSTR2 |
1-(1H-Benzoimidazol-2-ylmethyl)-3-{2-[(5-bromo-pyridin-2-yl)-(3,4-dichloro-benzyl)-amino]-ethyl}-thiourea |
300000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| SSTR2 |
1-{3-[(5-Bromo-pyridin-2-yl)-(3,4-dichloro-benzyl)-amino]-propyl}-3-[3-(pyridin-2-ylamino)-propyl]-thiourea |
300000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| SSTR2 |
1-{2-[(5-Bromo-pyridin-2-yl)-(3,4-dichloro-benzyl)-amino]-ethyl}-3-(4-piperidin-1-yl-phenyl)-thiourea |
300000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| SSTR2 |
1-{3-[(5-Bromo-pyridin-2-yl)-(3,4-dichloro-benzyl)-amino]-propyl}-3-(4-piperidin-1-yl-phenyl)-thiourea |
300000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| SSTR2 |
1-{3-[(4-Bromo-benzyl)-pyridin-2-yl-amino]-propyl}-3-[3-(pyridin-2-ylamino)-propyl]-thiourea |
114000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| SSTR2 |
1-{4-[(4-Bromo-benzyl)-pyridin-2-yl-amino]-butyl}-3-(3-phenyl-propyl)-thiourea |
300000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| SSTR2 |
1-(4-aminobutyl)-8-benzyl-12-[(2R)-2-hydroxypropyl]-4-[2-(1H-indol-3-yl)ethyl]-1,4,8,12-tetrazacyclopentadecane-2,5,9,13-tetrone |
176000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| SSTR2 |
1-(4-aminobutyl)-9-benzyl-13-[(2R)-2-hydroxypropyl]-5-[2-(1H-indol-3-yl)ethyl]-1,5,9,13-tetrazacyclohexadecane-2,6,10,14-tetrone |
198000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| SSTR2 |
methyl 3-[3-[3-[[2-[3-[acetyl(benzyl)amino]propanoyl-[2-(1H-indol-3-yl)ethyl]amino]acetyl]-(4-aminobutyl)amino]propanoyl-[(2R)-2-hydroxypropyl]amino]propanoyl-benzylamino]propanoate |
110000 |
NA |
NA |
NA |
NA |
NA |
TTD |