Support By : Li-lab
GENE_SYMBOL | DRUG_NAME | Ki (nM) | IC50 (nM) | Kd (nM) | EC50 (nM) | Potency (nM) | AC50 (nM) | Datasource |
---|---|---|---|---|---|---|---|---|
TACR3 | 7-Methoxy-2-phenyl-quinoline-4-carboxylic acid benzylamide | 533000 | NA | NA | NA | NA | NA | BindingDB |
TAS1R1 | Sodium 2-(4-methoxyphenoxy)propanoate | NA | NA|165000 | NA | 7900000|7000000|710000|840000|NA | NA | NA | PubChem |
TAS1R2 | Sodium 2-(4-methoxyphenoxy)propanoate | NA | 103000|168000|NA | NA | NA|24700000|31300000|600000|940000|118000 | NA | NA | PubChem |
TAS1R3 | Sodium 2-(4-methoxyphenoxy)propanoate | NA | NA|103000|168000|165000 | NA | 7900000|7000000|710000|840000|NA|24700000|31300000|600000|940000|118000 | NA | NA | PubChem |
TAS2R1 | Sucralose | NA | NA | NA | 36300000 | NA | NA | PubChem |
TAS2R13 | Potassium Chloride | NA | NA | NA | 5000000 | NA | NA | PubChem |
TAS2R14 | Vanillin | NA | NA | NA | 570000 | NA | NA | GtoPDB |
TAS2R14 | Potassium Chloride | NA | NA | NA | 5000000 | NA | NA | PubChem |
TAS2R14 | Coumestrol | NA | NA | NA | 358000 | NA | NA | GtoPDB |
TAS2R16 | 4-nitrophenyl-beta-D-mannopyranoside | NA | NA | NA | 650000 | NA | NA | GtoPDB |
TAS2R16 | Salicin | NA | NA | NA | 1400000 | NA | NA | GtoPDB |
TAS2R16 | Arbutin | NA | NA | NA | 5800000 | NA | NA | PubChem |
TAS2R16 | beta-Gentiobiose | NA | NA | NA | 3840000 | NA | NA | GtoPDB |
TAS2R16 | Probenecid | NA | 292000 | NA | NA | NA | NA | GtoPDB |
TAS2R16 | Phenyl beta-D-glucopyranoside | NA | NA | NA | 1100000 | NA | NA | GtoPDB |
TAS2R20 | Vanillin | NA | NA | NA | 530000 | NA | NA | GtoPDB |
TAS2R31 | Acesulfame potassium | NA | NA | NA | 3000000 | NA | NA | PubChem |
TAS2R31 | Acesulfame | NA | NA | NA | 2500000 | NA | NA | GtoPDB |
TAS2R31 | Potassium Chloride | NA | NA | NA | 5000000 | NA | NA | PubChem |
TAS2R31 | Saccharin | NA | NA | NA | 1100000|650000 | NA | NA | GtoPDB|PubChem |