GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
Slc6a11 |
2-[4-[(2,4-Dichlorobenzoyl)amino]piperidin-1-yl]acetic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
Slc6a11 |
N-(1-benzylpiperidin-4-yl)-2-methylpropanamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
Slc6a11 |
2,4-dichloro-N-(1-propylpiperidin-4-yl)benzamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
Slc6a11 |
2,4-dichloro-N-(1-ethylpiperidin-4-yl)benzamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
Slc6a11 |
N-(1-benzylpiperidin-4-yl)-3-(trifluoromethyl)benzamide |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
Slc6a11 |
CI-966 |
NA |
333000 |
NA |
NA |
NA |
NA |
TTD |
Slc6a11 |
Guvacine |
NA |
110000 |
NA |
NA |
NA |
NA |
TTD |
Slc6a11 |
N-(1-benzylpiperidin-4-yl)benzamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
Slc6a11 |
2,4-dichloro-N-piperidin-4-ylbenzamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
Slc6a11 |
Hinokinin |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
Slc6a11 |
Nipecotic Acid |
NA |
106000 |
NA |
NA |
NA |
NA |
TTD |
Slc6a11 |
2,4-dichloro-N-[1-(pyridin-2-ylmethyl)piperidin-4-yl]benzamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
Slc6a11 |
2-(2-Amino-2-thiazolin-4-yl)acetic acid |
NA |
125892.54 |
NA |
NA |
NA |
NA |
TTD |
Slc6a11 |
Tiagabine |
NA |
917000 |
NA |
NA |
NA |
NA |
TTD |
Slc6a11 |
2,4-dichloro-N-(1-methylpiperidin-4-yl)benzamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
Slc6a11 |
Nipecotic acid, S-(+)- |
NA |
2320000 |
NA |
NA |
NA |
NA |
TTD |
Slc6a11 |
N-(1-benzylpiperidin-4-yl)-4-fluorobenzamide |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
Slc6a11 |
(3S)-8-benzhydrylidene-1,2,3,4,6,7,9,9a-octahydroquinolizine-3-carboxylic acid |
NA |
876000 |
NA |
NA |
NA |
NA |
TTD |
Slc6a11 |
(3R,8R)-8-benzhydryl-2,3,4,6,7,8,9,9a-octahydro-1H-quinolizine-3-carboxylic acid |
NA |
2043000 |
NA |
NA |
NA |
NA |
TTD |
Slc6a11 |
(3S,8R)-8-benzhydryl-2,3,4,6,7,8,9,9a-octahydro-1H-quinolizine-3-carboxylic acid |
NA |
782000 |
NA |
NA |
NA |
NA |
TTD |