| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| TAS2R9 |
Pirenzepine |
NA |
NA |
NA |
1800000 |
NA |
NA |
GtoPDB |
| TAS2R9 |
Potassium Chloride |
NA |
NA |
NA |
5000000 |
NA |
NA |
PubChem |
| TAS2R9 |
Procainamide |
NA |
NA |
NA |
2800000 |
NA |
NA |
GtoPDB |
| TBK1 |
2-Amino-5-oxo-7-(4-oxocyclohexyl)chromeno[2,3-b]pyridine-3-carboxylic acid |
NA |
630957.34 |
NA |
NA |
NA |
NA |
TTD |
| TBK1 |
5-Amino-9-oxo-12-prop-1-en-2-yl-2-oxa-4,13-diazatricyclo[8.4.0.03,8]tetradeca-1(14),3,5,7,10,12-hexaene-6-carboxylic acid |
NA |
524807.46 |
NA |
NA |
NA |
NA |
TTD |
| TBXA2R |
5-[2-Imidazol-1-yl-1-phenyl-prop-(Z)-ylideneaminooxy]-pentanoic acid |
NA |
295000 |
NA |
NA |
NA |
NA |
TTD |
| TBXA2R |
Imipenem |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| TBXA2R |
5-[1-Phenyl-1-pyridazin-3-yl-meth-(E)-ylideneaminooxy]-pentanoic acid |
NA |
104000 |
NA |
NA |
NA |
NA |
TTD |
| TBXA2R |
(Z)-7-[(1R,2S,3R)-3-(hexylsulfanylmethyl)-7-oxabicyclo[2.2.1]heptan-2-yl]hept-5-enoic acid |
NA |
115000 |
NA |
NA |
NA |
NA |
TTD |
| TBXA2R |
1-(3,4,5-Trimethoxyanilino)-3,4-dihydroisoquinoline-6,7-diol |
120226.44 |
NA |
NA |
NA |
NA |
NA |
TTD |
| TBXA2R |
Cefazolin |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| TBXA2R |
Meropenem |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| TBXA2R |
(Z)-7-(3-heptylsulfanyl-7-oxabicyclo[2.2.1]heptan-2-yl)hept-5-enoic acid |
NA |
230000 |
NA |
NA |
NA |
NA |
TTD |
| TBXA2R |
(Z)-7-[3-(octylsulfanylmethyl)-7-oxabicyclo[2.2.1]heptan-2-yl]hept-5-enoic acid |
NA |
547000 |
NA |
NA |
NA |
NA |
TTD |
| TBXA2R |
2-(3-((1-(2,4-difluorobenzyl)-6-oxo-1,6-dihydropyridazin-3-yl)methyl)-5-fluoro-2-methyl-1H-indol-1-yl)acetic acid |
NA |
560000 |
NA |
NA |
NA |
NA |
TTD |
| TBXA2R |
Cefepime |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| TBXA2R |
Ceftazidime |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| TBXA2R |
Aztreonam |
NA |
NA |
NA |
NA |
NA |
400000 |
PubChem |
| TBXA2R |
Carumonam |
NA |
NA |
NA |
NA |
NA |
500000 |
PubChem |
| TBXA2R |
Doripenem |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |