| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| TBXAS1 |
(6-{2-[(E)-Phenyl-pyridin-4-yl-methoxyimino]-propyl}-5,6,7,8-tetrahydro-naphthalen-1-yloxy)-acetic acid |
NA |
210000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| TBXAS1 |
(6-{2-[(E)-Phenyl-pyridin-2-yl-methoxyimino]-propyl}-5,6,7,8-tetrahydro-naphthalen-1-yloxy)-acetic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| TBXAS1 |
2-[[5-[3-Oxo-3-(2-phenyl-2-pyridin-3-ylhydrazinyl)propyl]-5,6,7,8-tetrahydronaphthalen-1-yl]oxy]acetic acid |
NA |
940000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| TBXAS1 |
{6-[4-(Phenyl-pyridin-3-yl-methyl)-pyrazol-1-ylmethyl]-5,6,7,8-tetrahydro-naphthalen-1-yloxy}-acetic acid |
NA |
320000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| TBXAS1 |
(Z)-7-[(2S,3S)-3-[(E,3R)-3-hydroxyoct-1-enyl]-7-oxabicyclo[2.2.1]heptan-2-yl]hept-5-enoic acid |
NA |
770000 |
NA |
NA |
NA |
NA |
TTD |
| TBXAS1 |
(Z)-7-[(2S,3S)-3-[(E,3S)-3-hydroxyoct-1-enyl]-7-oxabicyclo[2.2.1]heptan-2-yl]hept-5-enoic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| TBXAS1 |
(Z)-7-[(2R,3R)-3-[(E,3R)-3-hydroxyoct-1-enyl]-7-oxabicyclo[2.2.1]heptan-2-yl]hept-5-enoic acid |
NA |
470000 |
NA |
NA |
NA |
NA |
TTD |
| TBXAS1 |
(Z)-7-[(2R,3R)-3-[(E,3S)-3-hydroxyoct-1-enyl]-7-oxabicyclo[2.2.1]heptan-2-yl]hept-5-enoic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| TBXAS1 |
(Z)-7-[(2R,3S)-3-[(E,3S)-3-hydroxyoct-1-enyl]-7-oxabicyclo[2.2.1]heptan-2-yl]hept-5-enoic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| TBXAS1 |
(Z)-7-[(2S,3R)-3-[(E,3S)-3-hydroxyoct-1-enyl]-7-oxabicyclo[2.2.1]heptan-2-yl]hept-5-enoic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| TBXAS1 |
(Z)-7-[(2R,3S)-3-[(E,3R)-3-hydroxyoct-1-enyl]-7-oxabicyclo[2.2.1]heptan-2-yl]hept-5-enoic acid |
NA |
560000 |
NA |
NA |
NA |
NA |
TTD |
| TBXAS1 |
(Z)-7-[(2S,3R)-3-[(E,3R)-3-hydroxyoct-1-enyl]-7-oxabicyclo[2.2.1]heptan-2-yl]hept-5-enoic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| TBXAS1 |
Nitrendipine |
NA |
1000000 |
NA |
NA |
NA |
NA |
PubChem |
| TBXAS1 |
4-(2-Chloro-3-trifluoromethyl-phenyl)-2-imidazol-1-ylmethyl-6-methyl-1,4-dihydro-pyridine-3,5-dicarboxylic acid 5-ethyl ester 3-methyl ester: (succinate) |
NA |
125000 |
NA |
NA |
NA |
NA |
BindingDB |
| TBXAS1 |
5-O-ethyl 3-O-methyl 6-(2-imidazol-1-ylethoxymethyl)-2-methyl-4-(3-nitrophenyl)-3,4-dihydropyridine-3,5-dicarboxylate |
NA |
115000 |
NA |
NA |
NA |
NA |
BindingDB |
| TBXAS1 |
5-Ethyl 3-methyl 2,6-dimethyl-4-(3-nitrophenyl)-3,4-dihydropyridine-3,5-dicarboxylate |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB |
| TBXAS1 |
Imidazole |
NA |
670000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| TCF4 |
2-(((2-(4-Ethylphenyl)-5-methyloxazol-4-yl)methyl)thio)-N-phenethylacetamide |
364710 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| TCF4 |
Pnu-74654 |
180990 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| TDO2 |
O-[cyclohexyl(phenyl)methyl]hydroxylamine;hydrochloride |
NA |
2770000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |