Navigator

      Support By : Li-lab

Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
AKR1C2 3-[1-(4-chlorobenzoyl)-5-methoxy-3-methylindol-2-yl]-2-methyl-N-methylsulfonylpropanamide NA 115800 NA NA NA NA BindingDB
AKR1C2 4-[Methyl(phenylsulfonyl)amino]benzoic acid 119000 NA NA NA NA NA BindingDB|ChEMBL
AKR1C2 2-(4-hydroxy-2-oxo-3H-1,3-thiazol-5-yl)-N-(2-hydroxyphenyl)acetamide NA|102800 205700|NA NA NA NA NA BindingDB
AKR1C3 3-(1H-benzimidazol-2-ylamino)benzoic acid 142000 NA NA NA NA NA BindingDB|ChEMBL|TTD
AKR1C3 N-[(6-oxo-1H-pyrimidin-4-yl)methyl]pyrazolo[1,5-a]pyridine-2-carboxamide 118000 NA NA NA NA NA ChEMBL|TTD
AKR1C3 3-[(2,6-Dimethylpyrimidin-4-yl)amino]-4-methylbenzoic acid 144000 NA NA NA NA NA BindingDB|ChEMBL|TTD
AKR1C3 2-[(3-methyl-1H-pyrazol-1-yl)methyl]quinoline-4-carboxylic acid 117000 NA NA NA NA NA BindingDB|ChEMBL|TTD
AKR1C3 3-{[(4-Methylphenyl)sulfonyl]amino}benzoic acid 111000 NA NA NA NA NA BindingDB|ChEMBL|TTD
AKR1C3 118000 NA NA NA NA NA BindingDB
AKR1C3 3-(Naphthalene-2-sulfonamido)propanoic acid 148000 NA NA NA NA NA BindingDB|ChEMBL|TTD
AKR1C3 (E)-3-(4-methylsulfonylphenyl)-2-phenylprop-2-enoic acid NA 139200 NA NA NA NA BindingDB|TTD
AKR1C3 Jasmonic Acid 162000 NA NA NA NA NA BindingDB
AKR1C3 Methyl Jasmonate 153000 NA NA NA NA NA BindingDB|TTD
AKR1C3 (2E)-3-(3-hydroxy-4-methoxyphenyl)-2-(3,4,5-trimethoxy phenyl)acrylic acid NA 121100 NA NA NA NA BindingDB|TTD
AKR1C3 4-Methoxybenzophenone NA 180000 NA NA NA NA BindingDB|TTD
AKR1C3 5-[(2,5-Dimethyl-3-furoyl)amino]-2-hydroxybenzoic acid 118000 NA NA NA NA NA BindingDB|ChEMBL|TTD
AKR1C3 (E)-3-(3,4-dimethoxyphenyl)-2-naphthalen-1-ylprop-2-enoic acid NA 127800 NA NA NA NA BindingDB|TTD
AKR1C3 4-[Methyl(phenylsulfonyl)amino]benzoic acid 148000 NA NA NA NA NA BindingDB|ChEMBL|TTD
AKR1C4 (E)-3-[3-(3-methylbut-2-enyl)-5-[(4-methylphenyl)methylcarbamoyl]phenyl]prop-2-enoic acid NA 145000 NA NA NA NA BindingDB
AKT1 7-(4-fluoroanilino)-1-[(1R,3R)-3-hydroxycyclopentyl]-3-(4-methoxyphenyl)-4H-pyrimido[4,5-d]pyrimidin-2-one NA 125000 NA NA NA NA TTD