| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| AKR1C1 |
Gliclazide |
NA |
300000 |
NA |
NA |
NA |
NA |
PubChem |
| AKR1C1 |
3-(Naphthalene-2-sulfonamido)propanoic acid |
103000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL |
| AKR1C1 |
3a-phenyl-3,4-dihydro-2H-pyrrolo[1,2-a]benzimidazol-1-one |
NA |
167200 |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL |
| AKR1C1 |
Indomethacin |
NA |
130000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
| AKR1C1 |
Jasmonic Acid |
106000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| AKR1C1 |
4-[Methyl(phenylsulfonyl)amino]benzoic acid |
124000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL |
| AKR1C1 |
4-{[2-(Aminocarbonyl)phenoxy]methyl}-5-methyl-2-furamide |
122000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL |
| AKR1C1 |
(E)-3-[3-(3-methylbut-2-enyl)-4-(3-phenylpropanoyloxy)phenyl]prop-2-enoic acid |
NA |
187000 |
NA |
NA |
NA |
NA |
BindingDB |
| AKR1C2 |
4-[[3,5-Bis(trifluoromethyl)phenyl]amino]-1,2-benzoxazol-3-one |
NA |
118550 |
NA |
NA |
NA |
NA |
BindingDB |
| AKR1C2 |
(E)-3-[3-(3-methylbut-2-enyl)-5-[[3-(trifluoromethoxy)phenyl]methylcarbamoyl]phenyl]prop-2-enoic acid |
NA |
129000 |
NA |
NA |
NA |
NA |
BindingDB |
| AKR1C2 |
(E)-3-[3-(3-methylbut-2-enyl)-5-[[4-(trifluoromethoxy)phenyl]methylcarbamoyl]phenyl]prop-2-enoic acid |
NA |
165000 |
NA |
NA |
NA |
NA |
BindingDB |
| AKR1C2 |
(E)-3-[3-[2-(4-fluorophenyl)ethylcarbamoyl]-5-(3-methylbut-2-enyl)phenyl]prop-2-enoic acid |
NA |
148000 |
NA |
NA |
NA |
NA |
BindingDB |
| AKR1C2 |
(E)-3-[3-[2-(4-methoxyphenyl)ethylcarbamoyl]-5-(3-methylbut-2-enyl)phenyl]prop-2-enoic acid |
NA |
136000 |
NA |
NA |
NA |
NA |
BindingDB |
| AKR1C2 |
N-[2-bromo-5-[(E)-2-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)ethenyl]phenyl]-3-phenylpropanamide |
NA |
109000 |
NA |
NA |
NA |
NA |
BindingDB |
| AKR1C2 |
3-[(3,4-dimethoxyphenyl)methyl]-5-hydroxy-N-[3-(trifluoromethyl)phenyl]triazole-4-carboxamide |
NA |
108130 |
NA |
NA |
NA |
NA |
BindingDB |
| AKR1C2 |
2-(2,4-dioxo-1,3-thiazolidin-5-yl)-N-(2-hydroxyphenyl)acetamide |
102800|NA |
NA|205700 |
NA |
NA |
NA |
NA |
ChEMBL |
| AKR1C2 |
Gliclazide |
NA |
1000000 |
NA |
NA |
NA |
NA |
PubChem |
| AKR1C2 |
Drupanin |
NA |
107000|108000|125893 |
NA |
NA |
NA |
NA |
BindingDB |
| AKR1C2 |
7-benzoyl-4,5-dihydro-1,4-benzoxazepin-3(2H)-one |
137000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL |
| AKR1C2 |
2-(3-Hydroxyphenyl)quinoline-4-carboxylic acid |
121000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL |