| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| JAK2 |
US10040781, Example 217 |
NA |
980000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
US10040781, Example 158 |
NA |
171000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
US10040781, Example 428 |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
2-(((3R,4S)-3-fluoro-1-((S)-2-hydroxypropanoyl)piperidin-4-yl)oxy)-5-(4-((4-((R)-pyrrolidin-2-yl)phenyl)amino)-1,3,5-triazin-2-yl)benzonitrile |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
US10040781, Example 564 |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
US10040781, Example 256 |
NA |
144000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
(R)-2-((1-(2-cyanoacetyl)pyrrolidin-3-yl)oxy)-5-(4-((4-(4-(oxetan-3-yl)piperazin-1-yl)phenyl)amino)-1,3,5-triazin-2-yl)benzonitrile |
NA |
292000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
US10040781, Example 425 |
NA |
590000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
5-(4-((4-(4-(Oxetan-3-yl)piperazin-1-yl)phenyl)amino)-1,3,5-triazin-2-yl)-2-(2-oxa-8-azaspiro[4.5]decan-8-yl)benzonitrile |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
US10040781, Example 612 |
NA |
607000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
2-(((3R,4S)-3-fluoro-1-(tetrahydrofuran-3-yl)piperidin-4-yl)oxy)-5-(4-((4-(4-(oxetan-3-yl)piperazin-1-yl)phenyl)amino)-1,3,5-triazin-2-yl)benzonitrile |
NA |
740000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
TBK1/IKKepsilon-IN-5 |
NA |
802000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
US10040781, Example 346 |
NA |
511000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
2-(((3R,4S)-3-fluoro-1-(oxetan-3-yl)piperidin-4-yl)oxy)-5-(4-((4-(4-(oxetan-3-yl)piperazin-1-yl)phenyl)amino)-1,3,5-triazin-2-yl)benzonitrile |
NA |
602000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
US10040781, Example 233 |
NA |
333000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
2-(((3R,4S)-1-(2-(1H-pyrazol-5-yl)acetyl)-3-fluoropiperidin-4-yl)oxy)-5-(4-((4-(4-(oxetan-3-yl)piperazin-1-yl)phenyl)amino)-1,3,5-triazin-2-yl)benzonitrile |
NA |
127000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
US10040781, Example 515 |
NA |
355000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
5-(4-((4-(4-acetylpiperazin-1-yl)phenyl)amino)-1,3,5-triazin-2-yl)-2-((tetrahydro-2H-pyran-4-yl)oxy)benzonitrile |
NA |
224000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
US10040781, Example 444 |
NA |
476000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
US10040781, Example 126 |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB |