| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| JAK2 |
US10040781, Example 467 |
NA |
171000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
US10040781, Example 385 |
NA |
888000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
US10040781, Example 553 |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
US10040781, Example 18 |
NA |
271000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
US10040781, Example 255 |
NA |
227000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
US10040781, Example 231 |
NA |
486000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
US10040781, Example 357 |
NA |
511000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
2-(((3R,4S)-3-fluoro-1-((2S,4S)-4-hydroxy-5-oxopyrrolidine-2-carbonyl)piperidin-4-yl)oxy)-5-(4-((4-(4-(oxetan-3-yl)piperazin-1-yl)phenyl)amino)-1,3,5-triazin-2-yl)benzonitrile |
NA |
450000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
2-((5,5-Difluoro-6-oxopiperidin-3-yl)oxy)-5-(4-((4-(4-(oxetan-3-yl)piperazin-1-yl)phenyl)amino)-1,3,5-triazin-2-yl)benzonitrile |
NA |
153000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
US10040781, Example 91 |
NA |
693000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
US10040781, Example 537 |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
US10040781, Example 536 |
NA |
101000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
US10040781, Example 353 |
NA |
944000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
US10040781, Example 232 |
NA |
128000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
(R)-4-((4-(3-cyano-4-((1-(2-hydroxyacetyl)pyrrolidin-3-yl)oxy)phenyl)-1,3,5-triazin-2-yl)amino)-N-isopropylbenzamide |
NA |
604000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
2-(((3R,4S)-3-fluoro-1-(3-hydroxypropanoyl)piperidin-4-yl)oxy)-5-(4-((3-methoxy-4-(4-(oxetan-3-yl)piperazin-1-yl)phenyl)amino)-1,3,5-triazin-2-yl)benzonitrile |
NA |
110000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
(3R,4S)-methyl 4-(2-cyano-4-(4-((4-(4-(oxetan-3-yl)piperazin-1-yl)phenyl)amino)-1,3,5-triazin-2-yl)phenoxy)-3-fluoropiperidine-1-carboxylate |
NA |
680000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
2-(((S)-3,3-difluoro-1-((S)-2-oxooxazolidine-4-carbonyl)piperidin-4-yl)oxy)-5-(4-((4-(4-(oxetan-3-yl)piperazin-1-yl)phenyl)amino)-1,3,5-triazin-2-yl)benzonitrile |
NA |
184000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
5-(4-((4-(4-(Oxetan-3-yl)piperazin-1-yl)phenyl)amino)-1,3,5-triazin-2-yl)-2-(7-oxa-2-azaspiro[3.5]nonan-2-yl)benzonitrile |
NA |
170000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
2-(((4S,5R)-5-fluoro-1-(3-hydroxypropanoyl)-3,3-dimethylpiperidin-4-yl)oxy)-5-(4-((4-(4-(oxetan-3-yl)piperazin-1-yl)phenyl)amino)-1,3,5-triazin-2-yl)benzonitrile |
NA |
102000 |
NA |
NA |
NA |
NA |
BindingDB |