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      Support By : Li-lab

Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
ACHE but-(2E)-en-1,4-diyl-1,1'-bis(4-carboxypyridinium) dibromide (18) NA 3870000 NA NA NA NA BindingDB
ACHE but-(2E)-en-1,4-diyl-1,1'-bis(4-methyloxycarbonylpyridinium) dibromide (19) NA 401000 NA NA NA NA BindingDB
ACHE but-(2E)-en-1,4-diyl-1,1'-bis(4-carbamoylpyridinium) dibromide (20) NA 1200000 NA NA NA NA BindingDB
ACHE 1-[(E)-4-pyridin-1-ium-1-ylbut-2-enyl]pyridin-1-ium;dibromide NA 2290000 NA NA NA NA TTD
ACHE 2-Carboxyl-3,4-dihydroquinazoline NA 344800 NA NA NA NA BindingDB
ACHE 2-[Methyl(methylsulfanyl)phosphoryl]oxypropane NA NA 1500000 NA NA NA BindingDB
ACHE 2-(4-iodophenoxy)-N-[3-(4-methylpiperazin-1-yl)propyl]acetamide NA 138000 NA NA NA NA BindingDB|TTD
ACHE 2,2-Dimethyl-3-[methyl(methylsulfanyl)phosphoryl]oxybutane NA 720000 NA NA NA NA BindingDB|TTD
ACHE Pralidoxime Iodide 180000 NA NA NA NA NA TTD
ACHE Asoxime cation NA 667800 NA NA NA NA TTD
ACHE Obidoxime NA 640000 NA NA NA NA TTD
ACHE Pyridine-2-aldoxime NA NA|560000 210000|400000|790000|NA NA NA NA BindingDB|TTD
ACHE Pegamine NA 155100 NA NA NA NA BindingDB
ACHE Pralidoxime Chloride NA 1000000|366000|NA|996000|1190000|1210000 NA|3159000|706000|215000|187300 NA NA NA PubChem
ACHE Discorhabdin L NA 158000 NA NA NA NA TTD
ACHE Pralidoxime cation, (Z)- NA 878000 NA NA NA NA GtoPDB
ACHE 2-(Isoquinolin-2-ium-2-ylmethyl)isoquinolin-2-ium;dibromide NA 654000 NA NA NA NA TTD
ACHE 1,1'-(Pentane-1,5-diyl)di(pyridin-1-ium) dibromide NA 1270000 NA NA NA NA TTD
ACHE Trimedoxime Bromide NA 167000 NA NA NA NA TTD
ACHE 1,2,4-Oxadiazole-5-carboxaldehyde,3-ME,oxime NA 1000000 NA NA NA NA TTD