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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
SIRT2 Ac-Orn(Ac)-Lys(CSNH2)(CSNH2)-Orn(Ac)-NH2 NA 159100 NA NA NA NA BindingDB|TTD
SIRT2 8-Phenyl-Nicotinamide Adenine Dinucleotide NA 123000 NA NA NA NA BindingDB
SIRT2 methyl (2S)-2-[[(2S)-2-acetamido-6-(ethanethioylamino)hexanoyl]amino]propanoate NA 862000 NA NA NA NA BindingDB|TTD
SIRT2 Ac-Lys(Ac)-Asu(NH2)(NH2)-Lys(Ac)-NH2 NA 190200 NA NA NA NA BindingDB|TTD
SIRT2 4-((4-(2,3-dihydro-1H-inden-2-yl)-5-hydroxy-4H-1,2,4-triazol-3-ylthio)methyl)-7-hydroxy-2H-chromen-2-one NA 300000 NA NA NA NA TTD
SIRT2 NA 103000|103400 NA NA NA NA BindingDB
SIRT2 alpha-((5-Nitro-2-furanyl)methylene)-1H-benzimidazole-2-acetonitrile NA 127200 NA NA NA NA BindingDB
SIRT2 4-(3-(2-Hydroxybenzamido)phenylamino)-4-oxobut-2-enoic acid NA 1000000 NA NA NA NA TTD
SIRT2 2-[4-[(E)-2-phenylethenyl]anilino]benzamide NA 300000 NA NA NA NA TTD
SIRT2 2-[4-[Benzoyl(methyl)amino]anilino]benzamide NA 300000 NA NA NA NA TTD
SIRT2 Lamivudine NA 167700 NA NA NA NA BindingDB
SIRT2 4-[4-(Furan-2-amido)benzamido]-2-hydroxybenzoic acid NA 482000 NA NA NA NA BindingDB|TTD
SIRT2 5-{3-[(Furan-2-carbonyl)-amino]-benzoylamino}-2-hydroxy-benzoic acid NA 751000 NA NA NA NA BindingDB|TTD
SIRT2 tert-butyl N-[4-[(4-cyanophenyl)carbamoylamino]-2,2-dimethyl-3,4-dihydrochromen-6-yl]carbamate NA 110200 NA NA NA NA BindingDB|TTD
SIRT2 Cinnamoyl tryptamine NA 173000 NA NA NA NA BindingDB|TTD
SIRT2 4-[(6-Bromo-2-hydroxynaphthalen-1-yl)methyl]-5-(4-methylphenyl)-1,2-dihydropyrazol-3-one NA 200000 NA NA NA NA TTD
SIRT2 4-[(2-Hydroxy-3-methoxynaphthalen-1-yl)methyl]-5-(4-methylphenyl)-1,2-dihydropyrazol-3-one NA 200000 NA NA NA NA TTD
SIRT2 NA 4500000 NA NA NA NA BindingDB
SIRT2 5-[4-(Furan-2-amido)benzamido]-2-hydroxybenzoic acid NA 453000 NA NA NA NA BindingDB|TTD
SIRT2 Niacinamide NA 100500 NA NA NA NA BindingDB|PubChem