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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
STAT3 2-Hydroxy-4-[[2-[(4-methylphenyl)sulfonyl-[(2-methylpropan-2-yl)oxycarbonyl]amino]acetyl]amino]benzoic acid NA 300000 NA NA NA NA TTD
STAT3 2-Hydroxy-4-[[2-[methyl-(4-methylphenyl)sulfonylamino]acetyl]amino]benzoic acid NA 300000 NA NA NA NA TTD
STAT3 Ac-Tyr(PO3H2)-Ser-Thr-Val-Val-His-NH2 NA 150000 NA NA NA NA TTD
STAT3 2-Hydroxy-5-(N-(4-methoxybenzyl)-4-phenoxybenzamido)benzoic acid NA 118100 NA NA NA NA TTD
STAT3 5-(N-Benzyl-2-(N,4-dimethylphenylsulfonamido)acetamido)-2-hydroxybenzoic acid NA 1000000 NA NA NA NA TTD
STAT3 5-[[2-[Benzyl-(4-phenylphenyl)sulfonylamino]acetyl]-[(4-piperidin-4-ylphenyl)methyl]amino]-2-hydroxybenzoic acid NA 300000 NA NA NA NA TTD
STAT3 5-(N-Benzyl-2-(N-benzyl-4-methylphenylsulfonamido)acetamido)-2-hydroxybenzoic acid NA 201300 NA NA NA NA TTD
STAT3 6-(3,4-dihydroxyphenyl)-8-hydroxy-1,3-dimethyl-4H-cyclohepta[c]furan-4-one NA 106000 NA NA NA NA TTD
STAT3 STAT5 Inhibitor NA 180000 NA NA NA NA TTD
STAT3 (2S)-2-[(2S)-2-[(4-cyanophenyl)formamido]-3-[4-(phosphonooxy)phenyl]propanamido]-4-methylpentanoic acid NA 310000 NA NA NA NA TTD
STING1 2-(7-methoxy-5,6-dimethyl-9-oxo-10H-acridin-4-yl)acetic acid NA NA NA 134290 NA NA BindingDB
STING1 2-[(6-Pyridazin-4-ylpyridazine-3-carbonyl)amino]-5-(trifluoromethyl)benzoic acid NA NA NA 1938000 NA NA BindingDB
STING1 Mangostin NA NA|137000 157000|NA|137000 NA NA NA PubChem
STK10 3-[(3-Chloro-4-methoxyphenyl)methylamino]-4-[2-(trifluoromethyl)phenyl]pyrrole-2,5-dione 130000 NA NA NA NA NA BindingDB
STK10 3-[(3-Chloro-4-methoxyphenyl)methylamino]-4-(2-chlorophenyl)pyrrole-2,5-dione 190000 NA NA NA NA NA BindingDB
STK10 3-[(3-Chloro-4-methoxyphenyl)methylamino]-4-(2-methoxyphenyl)pyrrole-2,5-dione 450000 NA NA NA NA NA BindingDB
STS 4-Bromophenyl Sulfamate NA 912000 NA NA NA NA BindingDB|TTD
STS 3-Nitrophenyl Sulfamate NA 120000 NA NA NA NA BindingDB|TTD
STS 4-Chlorophenyl Sulfamate NA 1580000|1584800|1585000 NA NA NA NA BindingDB|TTD
STS Sulfamic acid 3-iodophenyl ester NA 120000 NA NA NA NA BindingDB|TTD