| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| STS |
4-Formylphenyl sulfamate |
NA |
254000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| STS |
Sulfamic acid 4-acetyl-phenyl ester |
NA |
302000 |
NA |
NA |
NA |
NA |
BindingDB |
| STS |
[(8R,9S,13S,14S)-13-methyl-17-oxo-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthren-3-yl]methanesulfonic acid |
140000|600000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| STS |
3-Cyanophenyl sulfamate |
NA |
190500|191000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| STS |
4-Nitrophenyl sulfamate |
NA |
330000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| STS |
difluoro-[(8R,9S,13S,14S)-13-methyl-17-oxo-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthren-3-yl]methanesulfonic acid |
147000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| STS |
Phenylsulfamate |
NA |
10000000 |
NA |
NA |
NA |
NA |
TTD |
| STS |
(8R,9S,13S,14S)-13-Methyl-2-methylsulfanyl-17-oxo-7,8,9,11,12,13,14,15,16,17-decahydro-6H-cyclopenta[a]phenanthrene-3-sulfonic acid amide |
NA |
120000 |
NA |
NA |
NA |
NA |
BindingDB |
| STS |
[(8R,9S,13S,14S)-13-methyl-17-oxo-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthren-3-yl]methanesulfonamide |
350000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| STS |
3-[Amino-[(6-oxo-7,8,9,10-tetrahydrobenzo[c]chromen-3-yl)oxy]phosphinothioyl]oxy-7,8,9,10-tetrahydrobenzo[c]chromen-6-one |
NA |
109970 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| STS |
4-Methylphenyl sulfamate |
NA |
10000000 |
NA |
NA |
NA |
NA |
TTD |
| STS |
3-Chlorophenyl sulfamate |
NA |
537000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| STS |
(8R,9S,13S,14S)-3-hydroxy-13-methyl-17-oxo-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthrene-4-carboxylic acid |
NA |
215000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| STS |
Sulfamic acid, 2,2,2-trichloroethyl ester |
NA |
750000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| STS |
Sulfamic acid 4-[(E)-(3-phenyl-acryloyl)]-phenyl ester |
NA |
263000 |
NA |
NA |
NA |
NA |
BindingDB |
| STS |
Sulfamic acid 3-fluorophenyl ester |
NA |
2080000|2089000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| STS |
4-Fluorophenyl Sulfamate |
NA |
537000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| STS |
3-Bromophenyl sulfamate |
NA |
257000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| STS |
3-Methylphenyl sulfamate |
NA |
2080000|2089000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| STS |
4-Cyanophenyl sulfamate |
NA |
300000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |