| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| TDP1 |
N-[2-(5,11-dioxoindeno[1,2-c]isoquinolin-6-yl)ethyl]-4-methylbenzenesulfonamide |
NA |
111000 |
NA |
NA |
NA |
NA |
TTD |
| TDP1 |
N-[3-(5,11-dioxoindeno[1,2-c]isoquinolin-6-yl)propyl]-4-methylbenzenesulfonamide |
NA |
111000 |
NA |
NA |
NA |
NA |
TTD |
| TDP1 |
N-[4-(5,11-dioxoindeno[1,2-c]isoquinolin-6-yl)butyl]-4-methylbenzenesulfonamide |
NA |
111000 |
NA |
NA |
NA |
NA |
TTD |
| TDP1 |
N-[5-(5,11-dioxoindeno[1,2-c]isoquinolin-6-yl)pentyl]-4-methylbenzenesulfonamide |
NA |
111000 |
NA |
NA |
NA |
NA |
TTD |
| TDP1 |
N-[7-(5,11-dioxoindeno[1,2-c]isoquinolin-6-yl)heptyl]-4-methylbenzenesulfonamide |
NA |
111000 |
NA |
NA |
NA |
NA |
TTD |
| TDP1 |
N-[8-(5,11-dioxoindeno[1,2-c]isoquinolin-6-yl)octyl]-4-methylbenzenesulfonamide |
NA |
111000 |
NA |
NA |
NA |
NA |
TTD |
| TDP1 |
N-[9-(5,11-dioxoindeno[1,2-c]isoquinolin-6-yl)nonyl]-4-methylbenzenesulfonamide |
NA |
111000 |
NA |
NA |
NA |
NA |
TTD |
| TDP1 |
N-[10-(5,11-dioxoindeno[1,2-c]isoquinolin-6-yl)decyl]-4-methylbenzenesulfonamide |
NA |
111000 |
NA |
NA |
NA |
NA |
TTD |
| TDP1 |
N-[11-(5,11-dioxoindeno[1,2-c]isoquinolin-6-yl)undecyl]-4-methylbenzenesulfonamide |
NA |
111000 |
NA |
NA |
NA |
NA |
TTD |
| TDP1 |
N-[12-(5,11-dioxoindeno[1,2-c]isoquinolin-6-yl)dodecyl]-4-methylbenzenesulfonamide |
NA |
111000 |
NA |
NA |
NA |
NA |
TTD |
| TDP1 |
4-bromo-N-[2-(5,11-dioxoindeno[1,2-c]isoquinolin-6-yl)ethyl]benzenesulfonamide |
NA |
111000 |
NA |
NA |
NA |
NA |
TTD |
| TDP1 |
4-bromo-N-[3-(5,11-dioxoindeno[1,2-c]isoquinolin-6-yl)propyl]benzenesulfonamide |
NA |
111000 |
NA |
NA |
NA |
NA |
TTD |
| TDP1 |
4-bromo-N-[4-(5,11-dioxoindeno[1,2-c]isoquinolin-6-yl)butyl]benzenesulfonamide |
NA |
111000 |
NA |
NA |
NA |
NA |
TTD |
| TDP1 |
4-bromo-N-[5-(5,11-dioxoindeno[1,2-c]isoquinolin-6-yl)pentyl]benzenesulfonamide |
NA |
111000 |
NA |
NA |
NA |
NA |
TTD |
| TDP1 |
4-bromo-N-[6-(5,11-dioxoindeno[1,2-c]isoquinolin-6-yl)hexyl]benzenesulfonamide |
NA |
111000 |
NA |
NA |
NA |
NA |
TTD |
| TDP1 |
4-bromo-N-[7-(5,11-dioxoindeno[1,2-c]isoquinolin-6-yl)heptyl]benzenesulfonamide |
NA |
111000 |
NA |
NA |
NA |
NA |
TTD |
| TDP1 |
4-bromo-N-[8-(5,11-dioxoindeno[1,2-c]isoquinolin-6-yl)octyl]benzenesulfonamide |
NA |
111000 |
NA |
NA |
NA |
NA |
TTD |
| TDP1 |
4-bromo-N-[9-(5,11-dioxoindeno[1,2-c]isoquinolin-6-yl)nonyl]benzenesulfonamide |
NA |
111000 |
NA |
NA |
NA |
NA |
TTD |
| TDP1 |
4-bromo-N-[10-(5,11-dioxoindeno[1,2-c]isoquinolin-6-yl)decyl]benzenesulfonamide |
NA |
111000 |
NA |
NA |
NA |
NA |
TTD |
| TDP1 |
4-bromo-N-[11-(5,11-dioxoindeno[1,2-c]isoquinolin-6-yl)undecyl]benzenesulfonamide |
NA |
111000 |
NA |
NA |
NA |
NA |
TTD |