| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| TDP1 |
N-[7-(5,11-dioxoindeno[1,2-c]isoquinolin-6-yl)heptyl]methanesulfonamide |
NA |
111000 |
NA |
NA |
NA |
NA |
TTD |
| TDP1 |
N-[8-(5,11-dioxoindeno[1,2-c]isoquinolin-6-yl)octyl]methanesulfonamide |
NA |
111000 |
NA |
NA |
NA |
NA |
TTD |
| TDP1 |
N-[9-(5,11-dioxoindeno[1,2-c]isoquinolin-6-yl)nonyl]methanesulfonamide |
NA |
111000 |
NA |
NA |
NA |
NA |
TTD |
| TDP1 |
N-[10-(5,11-dioxoindeno[1,2-c]isoquinolin-6-yl)decyl]methanesulfonamide |
NA |
111000 |
NA |
NA |
NA |
NA |
TTD |
| TDP1 |
N-[11-(5,11-dioxoindeno[1,2-c]isoquinolin-6-yl)undecyl]methanesulfonamide |
NA |
111000 |
NA |
NA |
NA |
NA |
TTD |
| TDP1 |
N-[12-(5,11-dioxoindeno[1,2-c]isoquinolin-6-yl)dodecyl]methanesulfonamide |
NA |
111000 |
NA |
NA |
NA |
NA |
TTD |
| TDP1 |
N-[2-(5,11-dioxoindeno[1,2-c]isoquinolin-6-yl)ethyl]benzenesulfonamide |
NA |
111000 |
NA |
NA |
NA |
NA |
TTD |
| TDP1 |
N-[3-(5,11-dioxoindeno[1,2-c]isoquinolin-6-yl)propyl]benzenesulfonamide |
NA |
111000 |
NA |
NA |
NA |
NA |
TTD |
| TDP1 |
N-[4-(5,11-dioxoindeno[1,2-c]isoquinolin-6-yl)butyl]benzenesulfonamide |
NA |
111000 |
NA |
NA |
NA |
NA |
TTD |
| TDP1 |
N-[5-(5,11-dioxoindeno[1,2-c]isoquinolin-6-yl)pentyl]benzenesulfonamide |
NA |
111000 |
NA |
NA |
NA |
NA |
TTD |
| TDP1 |
N-[6-(5,11-dioxoindeno[1,2-c]isoquinolin-6-yl)hexyl]benzenesulfonamide |
NA |
111000 |
NA |
NA |
NA |
NA |
TTD |
| TDP1 |
N-[7-(5,11-dioxoindeno[1,2-c]isoquinolin-6-yl)heptyl]benzenesulfonamide |
NA |
111000 |
NA |
NA |
NA |
NA |
TTD |
| TDP1 |
N-[8-(5,11-dioxoindeno[1,2-c]isoquinolin-6-yl)octyl]benzenesulfonamide |
NA |
111000 |
NA |
NA |
NA |
NA |
TTD |
| TDP1 |
N-[9-(5,11-dioxoindeno[1,2-c]isoquinolin-6-yl)nonyl]benzenesulfonamide |
NA |
111000 |
NA |
NA |
NA |
NA |
TTD |
| TDP1 |
N-[6-(3-aminopropyl)-11-hydroxy-5-oxo-11H-indeno[1,2-c]isoquinolin-3-yl]acetamide |
NA |
111000 |
NA |
NA |
NA |
NA |
TTD |
| TDP1 |
N-[6-(3-hydroxypropyl)-5,11-dioxoindeno[1,2-c]isoquinolin-3-yl]acetamide |
NA |
111000 |
NA |
NA |
NA |
NA |
TTD |
| TDP1 |
N-[6-(3-azidopropyl)-5,11-dioxoindeno[1,2-c]isoquinolin-3-yl]acetamide |
NA |
111000 |
NA |
NA |
NA |
NA |
TTD |
| TDP1 |
6-(3-Hydroxypropyl)-3-nitroindeno[1,2-c]isoquinoline-5,11-dione |
NA |
111000 |
NA |
NA |
NA |
NA |
TTD |
| TDP1 |
(E)-2-cyano-3-naphthalen-2-ylprop-2-enethioamide |
NA |
333000 |
NA |
NA |
NA |
NA |
TTD |
| TDP1 |
(Z)-4-((2,4-dioxothiazolidin-5-ylidene)methyl)benzoic acid |
NA |
111000 |
NA |
NA |
NA |
NA |
TTD |