| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| TDP2 |
7-phenyl-1H-quinazoline-2,4-dione |
NA |
111000 |
NA |
NA |
NA |
NA |
TTD |
| TDP2 |
(2-Cyanophenyl) 2-methyl-4,9-dioxofuro[2,3-g]quinoline-3-carboxylate |
NA |
111000 |
NA |
NA |
NA |
NA |
TTD |
| TDP2 |
N-(4-methoxyphenyl)-2-methyl-4,9-dioxofuro[2,3-g]quinoline-3-carboxamide |
NA |
111000 |
NA |
NA |
NA |
NA |
TTD |
| TDP2 |
N-ethyl-2-methyl-4,9-dioxofuro[2,3-g]quinoline-3-carboxamide |
NA |
111000 |
NA |
NA |
NA |
NA |
TTD |
| TDP2 |
N-(3-chlorophenyl)-2-methyl-4,9-dioxofuro[2,3-g]quinoline-3-carboxamide |
NA |
111000 |
NA |
NA |
NA |
NA |
TTD |
| TDP2 |
N-(2-hydroxyphenyl)-2-methyl-4,9-dioxofuro[2,3-g]quinoline-3-carboxamide |
NA |
111000 |
NA |
NA |
NA |
NA |
TTD |
| TDP2 |
Naphthalen-2-yl 2-methyl-4,9-dioxofuro[2,3-g]quinoline-3-carboxylate |
NA |
111000 |
NA |
NA |
NA |
NA |
TTD |
| TDP2 |
ethyl 4,9-dioxo-2H-pyrazolo[3,4-g]quinoline-3-carboxylate |
NA |
111000 |
NA |
NA |
NA |
NA |
TTD |
| TDP2 |
2-methyl-4,9-dioxo-N-phenylfuro[2,3-g]quinoline-3-carboxamide |
NA |
111000 |
NA |
NA |
NA |
NA |
TTD |
| TDP2 |
Ethyl 1,2-dimethyl-4,9-dioxopyrrolo[3,2-g]quinoline-3-carboxylate |
NA |
111000 |
NA |
NA |
NA |
NA |
TTD |
| TDP2 |
1,3-Benzodioxol-5-yl 2-methyl-4,9-dioxofuro[2,3-g]quinoline-3-carboxylate |
NA |
111000 |
NA |
NA |
NA |
NA |
TTD |
| TDP2 |
6-[(2S)-2,3-dihydroxypropyl]-3-iodoindeno[1,2-c]isoquinoline-5,11-dione |
NA |
111000 |
NA |
NA |
NA |
NA |
TTD |
| TDP2 |
6-(3-Morpholin-4-ylpropyl)indeno[1,2-c][2,7]naphthyridine-5,11-dione |
NA |
111000 |
NA |
NA |
NA |
NA |
TTD |
| TDP2 |
6-(3-Imidazol-1-ylpropyl)indeno[1,2-c][2,7]naphthyridine-5,11-dione |
NA |
111000 |
NA |
NA |
NA |
NA |
TTD |
| TDP2 |
5-(furan-2-yl)-4H-isoquinoline-1,3-dione |
NA |
111000 |
NA |
NA |
NA |
NA |
TTD |
| TDP2 |
7-(3-aminophenyl)-4H-isoquinoline-1,3-dione |
NA |
111000 |
NA |
NA |
NA |
NA |
TTD |
| TDP2 |
6-benzyl-4H-isoquinoline-1,3-dione |
NA |
111000 |
NA |
NA |
NA |
NA |
TTD |
| TDP2 |
2-(1,3-dioxo-4H-isoquinolin-6-yl)benzoic acid |
NA |
111000 |
NA |
NA |
NA |
NA |
TTD |
| TDP2 |
6-(3-phenylphenyl)-4H-isoquinoline-1,3-dione |
NA |
111000 |
NA |
NA |
NA |
NA |
TTD |
| TDP2 |
6-(Furan-2-yl)benzo[de]isoquinoline-1,3-dione |
NA |
111000 |
NA |
NA |
NA |
NA |
TTD |