GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
TDP2 |
(4-Benzoylphenyl) 2-methyl-4,9-dioxofuro[2,3-g]quinoline-3-carboxylate |
NA |
111000 |
NA |
NA |
NA |
NA |
TTD |
TDP2 |
3-Dimethoxyphosphoryl-2-methylfuro[2,3-g]quinoline-4,9-dione |
NA |
111000 |
NA |
NA |
NA |
NA |
TTD |
TDP2 |
3,7-Dimethylfuro[2,3-g]quinoline-4,9-dione |
NA |
111000 |
NA |
NA |
NA |
NA |
TTD |
TDP2 |
N-ethyl-2-methyl-4,9-dioxofuro[3,2-g]quinoline-3-carboxamide |
NA |
111000 |
NA |
NA |
NA |
NA |
TTD |
TDP2 |
3-Acetyl-2-methylfuro[3,2-g]quinoline-4,9-dione |
NA |
111000 |
NA |
NA |
NA |
NA |
TTD |
TDP2 |
(4E)-4-[(3-bromo-4-methoxyphenyl)methylidene]-5-methyl-2-phenyl-3-pyrazolone |
NA |
102217 |
NA |
NA |
NA |
NA |
BindingDB |
TDP2 |
(2S)-3-(4-hydroxyphenyl)-2-[4-[3-[1-[(1S)-1-(1H-indol-3-ylmethyl)-2-keto-2-methoxy-ethyl]triazol-4-yl]-5-(piperazine-1-carbonyl)phenyl]triazol-1-yl]propionic acid |
NA |
128332 |
NA |
NA |
NA |
NA |
BindingDB |
TDP2 |
Sennoside A, analytical standard |
NA |
128309 |
NA |
NA |
NA |
NA |
BindingDB |
TDP2 |
5-[(E)-[1-(3,4-dimethylphenyl)-3-methyl-5-oxidanylidene-pyrazol-4-ylidene]methyl]-1,3-dimethyl-benzimidazol-2-one |
NA |
128314 |
NA |
NA |
NA |
NA |
BindingDB |
TDP2 |
10-(4-Chlorophenyl)[1,3]thiazolo[3,2-a]perimidine |
NA |
128357 |
NA |
NA |
NA |
NA |
BindingDB |
TDP2 |
2-[(5-Bromo-furan-2-carbonyl)-amino]-1-butyl-1H-pyrrolo[2,3-b]quinoxaline-3-carboxylic acid ethyl ester |
NA |
128305 |
NA |
NA |
NA |
NA |
BindingDB |
TDP2 |
N-(1-butyl-3-cyano-1H-pyrrolo[2,3-b]quinoxalin-2-yl)benzamide |
NA |
128345 |
NA |
NA |
NA |
NA |
BindingDB |
TDP2 |
1-Butyl-2-(toluene-4-sulfonylamino)-1H-pyrrolo[2,3-b]quinoxaline-3-carboxylic acid ethyl ester |
NA |
128345 |
NA |
NA |
NA |
NA |
BindingDB |
TDP2 |
2,4-Dibromo-6-[(quinolin-8-ylamino)methyl]phenol |
NA |
128357 |
NA |
NA |
NA |
NA |
BindingDB |
TDP2 |
3,6-Diamino-10-methylacridinium |
NA |
128332 |
NA |
NA |
NA |
NA |
BindingDB |
TDP2 |
2-furancarboxylic acid [2-ethoxy-4-[(E)-(3-methyl-5-oxo-1-phenyl-4-pyrazolylidene)methyl]phenyl] ester |
NA |
119078 |
NA |
NA |
NA |
NA |
BindingDB |
TDP2 |
2-N-cyclohexyl-1-N-(6-methoxyquinolin-8-yl)butane-1,2-diamine |
NA |
113281 |
NA |
NA |
NA |
NA |
BindingDB |
TDP2 |
Isopropyl-[3-[(6-methoxy-4-methyl-8-quinolyl)amino]propyl]amine |
NA |
128422 |
NA |
NA |
NA |
NA |
BindingDB |
TDP2 |
1-(4-Chlorophenyl)-3-isoquinolin-5-ylthiourea |
NA |
130127 |
NA |
NA |
NA |
NA |
BindingDB |
TDP2 |
Camptothecin |
NA |
111000 |
NA |
NA |
NA |
NA |
PubChem |