GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
TDP2 |
5-Bromo-6-methoxyquinolin-8-amine |
NA |
128315 |
NA |
NA |
NA |
NA |
BindingDB |
TDP2 |
(2-Chlorophenyl)-pyridin-2-yldiazene |
NA |
128126 |
NA |
NA |
NA |
NA |
BindingDB |
TDP2 |
N-[4-(dimethylamino)-1-methylindazol-3-yl]-1-methylimidazole-4-sulfonamide |
NA |
106216 |
NA |
NA |
NA |
NA |
BindingDB |
TDP2 |
GNF-Pf-4576 |
NA |
128329 |
NA |
NA |
NA |
NA |
BindingDB |
TDP2 |
Ethyl 3-(4-methylbenzyl)-1,4-dioxo-1,4-dihydro-2-naphthalenecarboxylate |
NA |
128305 |
NA |
NA |
NA |
NA |
BindingDB |
TDP2 |
2-[(4-Acetylphenyl)amino]-3-(4-morpholinyl)naphthoquinone |
NA |
128345 |
NA |
NA |
NA |
NA |
BindingDB |
TDP2 |
(6,7-Dimethoxy-1-isoquinolinyl)(4,5-dimethoxy-2-nitrophenyl)methanone |
NA |
128306 |
NA |
NA |
NA |
NA |
BindingDB |
TDP2 |
4-Bromonaphthalene-1,8-dicarboximide |
NA |
111000 |
NA |
NA |
NA |
NA |
TTD |
TDP2 |
2-(1,1-dioxothiolan-3-yl)-5-methyl-1H-pyrazol-3-one |
NA |
128284 |
NA |
NA |
NA |
NA |
BindingDB |
TDP2 |
2-Anilino-3-piperidin-1-ylnaphthalene-1,4-dione |
NA |
128324 |
NA |
NA |
NA |
NA |
BindingDB |
TDP2 |
2-[5-[Bis(3-methyl-5-oxo-1,2-dihydropyrazol-4-yl)methyl]furan-2-yl]benzoic acid |
NA |
128318 |
NA |
NA |
NA |
NA |
BindingDB |
TDP2 |
3-[5-[Bis(3-methyl-5-oxo-1,2-dihydropyrazol-4-yl)methyl]furan-2-yl]benzoic acid |
NA |
128325 |
NA |
NA |
NA |
NA |
BindingDB |
TDP2 |
3-[5-[Bis(3-methyl-5-oxo-1,2-dihydropyrazol-4-yl)methyl]-2-furanyl]benzoic acid methyl ester |
NA |
128332 |
NA |
NA |
NA |
NA |
BindingDB |
TDP2 |
2,3-bis(furan-2-yl)-N-(3-hydroxypropyl)quinoxaline-6-carboxamide |
NA |
128325 |
NA |
NA |
NA |
NA |
BindingDB |
TDP2 |
1-(1,3-Dioxolan-2-yl)-4-methylisoquinolin-5-amine |
NA |
128550 |
NA |
NA |
NA |
NA |
BindingDB |
TDP2 |
2-(4-methoxyphenyl)-5-methyl-1,2-dihydro-3H-pyrazol-3-one |
NA |
128216 |
NA |
NA |
NA |
NA |
BindingDB |
TDP2 |
2-Benzenesulfonylamino-1-butyl-1H-pyrrolo[2,3-b]quinoxaline-3-carboxylic acid ethyl ester |
NA |
128325 |
NA |
NA |
NA |
NA |
BindingDB |
TDP2 |
4-(4-Ethoxyanilino)-1,2-naphthalenedione |
NA |
128460 |
NA |
NA |
NA |
NA |
BindingDB |
TDP2 |
10-[3-(Diethylamino)propylamino]-5-hydroxy-1,14-diazatetracyclo[7.6.1.02,7.013,16]hexadeca-2(7),3,5,9,11,13(16),14-heptaen-8-one;hydrochloride |
NA |
128383 |
NA |
NA |
NA |
NA |
BindingDB |
TDP2 |
5-Methyl-3-(methylamino)phenazin-5-ium |
NA |
128357 |
NA |
NA |
NA |
NA |
BindingDB |