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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
TDP2 5-Bromo-6-methoxyquinolin-8-amine NA 128315 NA NA NA NA BindingDB
TDP2 (2-Chlorophenyl)-pyridin-2-yldiazene NA 128126 NA NA NA NA BindingDB
TDP2 N-[4-(dimethylamino)-1-methylindazol-3-yl]-1-methylimidazole-4-sulfonamide NA 106216 NA NA NA NA BindingDB
TDP2 GNF-Pf-4576 NA 128329 NA NA NA NA BindingDB
TDP2 Ethyl 3-(4-methylbenzyl)-1,4-dioxo-1,4-dihydro-2-naphthalenecarboxylate NA 128305 NA NA NA NA BindingDB
TDP2 2-[(4-Acetylphenyl)amino]-3-(4-morpholinyl)naphthoquinone NA 128345 NA NA NA NA BindingDB
TDP2 (6,7-Dimethoxy-1-isoquinolinyl)(4,5-dimethoxy-2-nitrophenyl)methanone NA 128306 NA NA NA NA BindingDB
TDP2 4-Bromonaphthalene-1,8-dicarboximide NA 111000 NA NA NA NA TTD
TDP2 2-(1,1-dioxothiolan-3-yl)-5-methyl-1H-pyrazol-3-one NA 128284 NA NA NA NA BindingDB
TDP2 2-Anilino-3-piperidin-1-ylnaphthalene-1,4-dione NA 128324 NA NA NA NA BindingDB
TDP2 2-[5-[Bis(3-methyl-5-oxo-1,2-dihydropyrazol-4-yl)methyl]furan-2-yl]benzoic acid NA 128318 NA NA NA NA BindingDB
TDP2 3-[5-[Bis(3-methyl-5-oxo-1,2-dihydropyrazol-4-yl)methyl]furan-2-yl]benzoic acid NA 128325 NA NA NA NA BindingDB
TDP2 3-[5-[Bis(3-methyl-5-oxo-1,2-dihydropyrazol-4-yl)methyl]-2-furanyl]benzoic acid methyl ester NA 128332 NA NA NA NA BindingDB
TDP2 2,3-bis(furan-2-yl)-N-(3-hydroxypropyl)quinoxaline-6-carboxamide NA 128325 NA NA NA NA BindingDB
TDP2 1-(1,3-Dioxolan-2-yl)-4-methylisoquinolin-5-amine NA 128550 NA NA NA NA BindingDB
TDP2 2-(4-methoxyphenyl)-5-methyl-1,2-dihydro-3H-pyrazol-3-one NA 128216 NA NA NA NA BindingDB
TDP2 2-Benzenesulfonylamino-1-butyl-1H-pyrrolo[2,3-b]quinoxaline-3-carboxylic acid ethyl ester NA 128325 NA NA NA NA BindingDB
TDP2 4-(4-Ethoxyanilino)-1,2-naphthalenedione NA 128460 NA NA NA NA BindingDB
TDP2 10-[3-(Diethylamino)propylamino]-5-hydroxy-1,14-diazatetracyclo[7.6.1.02,7.013,16]hexadeca-2(7),3,5,9,11,13(16),14-heptaen-8-one;hydrochloride NA 128383 NA NA NA NA BindingDB
TDP2 5-Methyl-3-(methylamino)phenazin-5-ium NA 128357 NA NA NA NA BindingDB