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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
TDP2 NA 128332 NA NA NA NA BindingDB
TDP2 Vanadate(3-) NA 40000000 NA NA NA NA BindingDB|TTD
TDP2 4-[(3-Chloro-1-benzothiophen-2-yl)methylideneamino]phenol NA 128305 NA NA NA NA BindingDB
TDP2 3-Amino-4-(furan-2-yl)-6-phenylthieno[2,3-b]pyridine-2-carbonitrile NA 128320 NA NA NA NA BindingDB
TDP2 (4-Amino-1,2,4-triazol-3-yl)-[[5-(2-nitrophenyl)-2-furyl]methyleneamino]amine NA 128345 NA NA NA NA BindingDB
TDP2 2-chloro-N-(3-cyano-1-prop-2-enylpyrrolo[3,2-b]quinoxalin-2-yl)benzamide NA 128310 NA NA NA NA BindingDB
TDP2 N-[3-cyano-1-(4-methoxyphenyl)pyrrolo[3,2-b]quinoxalin-2-yl]furan-2-carboxamide NA 128225 NA NA NA NA BindingDB
TDP2 Ethyl 1-butyl-2-(furan-2-carbonylamino)pyrrolo[3,2-b]quinoxaline-3-carboxylate NA 128300 NA NA NA NA BindingDB
TDP2 1,3-Dioxo-1,2,3,4-tetrahydro-isoquinoline-6-carboxylic acid NA 111000 NA NA NA NA TTD
TDP2 N-(4-hydroxynaphthalen-1-yl)thiophene-2-sulfonamide NA 128486 NA NA NA NA BindingDB
TDP2 N-[4-(3,4-dimethoxyphenyl)thiophen-2-yl]-1-methyl-6-oxo-5-phenylmethoxypyrimidine-4-carboxamide NA NA NA 150000 NA NA TTD
TDP2 [1-[4-(3,4-Dimethoxyphenyl)thiophene-2-carbonyl]piperidin-3-yl]-dimethoxyphosphorylmethanone NA NA NA 150000 NA NA TTD
TDP2 3-[4-(3,4-dimethoxyphenyl)thiophen-2-yl]-N-methylsulfonylbenzamide NA NA NA 150000 NA NA TTD
TDP2 4-[4-(3,4-dimethoxyphenyl)thiophen-2-yl]-N-methylsulfonylbenzamide NA NA NA 150000 NA NA TTD
TDP2 2-(naphthalen-1-yl)-2H-benzo[d][1,2,3]triazol-5-amine NA 128306 NA NA NA NA BindingDB
TDP2 N-(2,1,3-benzothiadiazol-5-yl)pyrrolidine-1-carbothioamide NA 128332 NA NA NA NA BindingDB
TDP2 (2Z)-2-[(5-methylfuran-2-yl)methylidene]-1,3-dioxoindene-5-carboxylic acid NA 128332 NA NA NA NA BindingDB
TDP2 N-(2,1,3-benzothiadiazol-5-yl)azepane-1-carbothioamide NA 128315 NA NA NA NA BindingDB
TDP2 N-2,1,3-benzothiadiazol-5-yl-1-piperidinecarbothioamide NA 128370 NA NA NA NA BindingDB
TDP2 3-tert-butyl-1-phenyl-1H-pyrazol-5-ol NA 128345 NA NA NA NA BindingDB