GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
TDP2 |
|
NA |
128332 |
NA |
NA |
NA |
NA |
BindingDB |
TDP2 |
Vanadate(3-) |
NA |
40000000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
TDP2 |
4-[(3-Chloro-1-benzothiophen-2-yl)methylideneamino]phenol |
NA |
128305 |
NA |
NA |
NA |
NA |
BindingDB |
TDP2 |
3-Amino-4-(furan-2-yl)-6-phenylthieno[2,3-b]pyridine-2-carbonitrile |
NA |
128320 |
NA |
NA |
NA |
NA |
BindingDB |
TDP2 |
(4-Amino-1,2,4-triazol-3-yl)-[[5-(2-nitrophenyl)-2-furyl]methyleneamino]amine |
NA |
128345 |
NA |
NA |
NA |
NA |
BindingDB |
TDP2 |
2-chloro-N-(3-cyano-1-prop-2-enylpyrrolo[3,2-b]quinoxalin-2-yl)benzamide |
NA |
128310 |
NA |
NA |
NA |
NA |
BindingDB |
TDP2 |
N-[3-cyano-1-(4-methoxyphenyl)pyrrolo[3,2-b]quinoxalin-2-yl]furan-2-carboxamide |
NA |
128225 |
NA |
NA |
NA |
NA |
BindingDB |
TDP2 |
Ethyl 1-butyl-2-(furan-2-carbonylamino)pyrrolo[3,2-b]quinoxaline-3-carboxylate |
NA |
128300 |
NA |
NA |
NA |
NA |
BindingDB |
TDP2 |
1,3-Dioxo-1,2,3,4-tetrahydro-isoquinoline-6-carboxylic acid |
NA |
111000 |
NA |
NA |
NA |
NA |
TTD |
TDP2 |
N-(4-hydroxynaphthalen-1-yl)thiophene-2-sulfonamide |
NA |
128486 |
NA |
NA |
NA |
NA |
BindingDB |
TDP2 |
N-[4-(3,4-dimethoxyphenyl)thiophen-2-yl]-1-methyl-6-oxo-5-phenylmethoxypyrimidine-4-carboxamide |
NA |
NA |
NA |
150000 |
NA |
NA |
TTD |
TDP2 |
[1-[4-(3,4-Dimethoxyphenyl)thiophene-2-carbonyl]piperidin-3-yl]-dimethoxyphosphorylmethanone |
NA |
NA |
NA |
150000 |
NA |
NA |
TTD |
TDP2 |
3-[4-(3,4-dimethoxyphenyl)thiophen-2-yl]-N-methylsulfonylbenzamide |
NA |
NA |
NA |
150000 |
NA |
NA |
TTD |
TDP2 |
4-[4-(3,4-dimethoxyphenyl)thiophen-2-yl]-N-methylsulfonylbenzamide |
NA |
NA |
NA |
150000 |
NA |
NA |
TTD |
TDP2 |
2-(naphthalen-1-yl)-2H-benzo[d][1,2,3]triazol-5-amine |
NA |
128306 |
NA |
NA |
NA |
NA |
BindingDB |
TDP2 |
N-(2,1,3-benzothiadiazol-5-yl)pyrrolidine-1-carbothioamide |
NA |
128332 |
NA |
NA |
NA |
NA |
BindingDB |
TDP2 |
(2Z)-2-[(5-methylfuran-2-yl)methylidene]-1,3-dioxoindene-5-carboxylic acid |
NA |
128332 |
NA |
NA |
NA |
NA |
BindingDB |
TDP2 |
N-(2,1,3-benzothiadiazol-5-yl)azepane-1-carbothioamide |
NA |
128315 |
NA |
NA |
NA |
NA |
BindingDB |
TDP2 |
N-2,1,3-benzothiadiazol-5-yl-1-piperidinecarbothioamide |
NA |
128370 |
NA |
NA |
NA |
NA |
BindingDB |
TDP2 |
3-tert-butyl-1-phenyl-1H-pyrazol-5-ol |
NA |
128345 |
NA |
NA |
NA |
NA |
BindingDB |