| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| TDP2 |
N-cyclohexyl-6-methyl-2-pyridin-3-ylimidazo[1,2-a]pyridin-3-amine |
NA |
128238 |
NA |
NA |
NA |
NA |
BindingDB |
| TDP2 |
N-[(2-pyrrolidin-1-ylphenyl)carbamothioyl]furan-2-carboxamide |
NA |
128320 |
NA |
NA |
NA |
NA |
BindingDB |
| TDP2 |
2-[2-[2-[[3-[(4-Chlorophenyl)methoxy]-4-methoxyphenyl]methylidene]hydrazinyl]-4-oxo-5-thiazolyl]acetic acid |
NA |
128324 |
NA |
NA |
NA |
NA |
BindingDB |
| TDP2 |
(6E)-6-[[2-(4-azanyl-5-methyl-1,2,4-triazol-3-yl)hydrazinyl]methylidene]cyclohexa-2,4-dien-1-one |
NA |
128345 |
NA |
NA |
NA |
NA |
BindingDB |
| TDP2 |
10-(4-Methylphenyl)-7-nitropyrimido[4,5-b]quinoline-2,4-dione |
NA |
128332 |
NA |
NA |
NA |
NA |
BindingDB |
| TEAD1 |
2-chloro-N-{2-[(4-chlorophenyl)thio]ethyl}acetamide |
NA |
182000 |
NA |
NA |
NA |
NA |
BindingDB |
| TEAD4 |
2-((3-Bromophenyl)amino)benzoic acid |
NA |
NA |
234000 |
NA |
NA |
NA |
BindingDB |
| TEC |
N-(3-fluorobenzyl)quinolin-2-amine |
NA |
NA |
177000 |
NA |
NA |
NA |
BindingDB |
| TEC |
N-benzylquinolin-2-amine |
NA |
NA |
193000 |
NA |
NA |
NA |
BindingDB |
| TEC |
3-(Quinolin-2-ylaminomethyl)-phenol |
NA |
NA |
234000 |
NA |
NA |
NA |
BindingDB |
| TEC |
N-(2-fluorobenzyl)quinolin-2-amine |
NA |
NA |
208000 |
NA |
NA |
NA |
BindingDB |
| TEC |
Staurosporine |
NA |
128000 |
NA |
NA |
NA |
NA |
BindingDB |
| TEC |
4-((Quinolin-2-ylamino)methyl)phenol |
NA |
NA |
292000 |
NA |
NA |
NA |
BindingDB |
| TEC |
N-((1H-pyrrol-2-yl)methyl)quinolin-2-amine |
NA |
NA |
285000 |
NA |
NA |
NA |
BindingDB |
| TEK |
Staurosporine |
NA |
59500000 |
NA |
NA |
NA |
NA |
BindingDB |
| TEK |
N-(4-methoxybenzyl)benzofuro[2,3-b]pyridin-4-amine |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| TEK |
4-Phenyl-[1]benzofuro[2,3-b]pyridine-3,6-diol |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| TEK |
(2R)-2-({[(9H-fluoren-9-yl)methoxy]carbonyl}amino)-3-(2-fluorophenyl)propanoic acid |
NA |
NA |
120000 |
NA |
NA |
NA |
BindingDB |
| TERF2 |
Ac-Leu-Ala-Leu-Lys-Tyr-Leu-OH |
461000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| TERF2 |
(3S,6S,9S,17S,20S)-9-amino-N,N,3-trimethyl-6-(2-methylpropyl)-2,5,8,19-tetraoxo-1,4,7,18-tetrazabicyclo[18.3.0]tricosane-17-carboxamide |
115000 |
NA |
NA |
NA |
NA |
NA |
TTD |