| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| TERT |
3-Diethylamino-N-[7-(3-diethylamino-propionylamino)-9-oxo-9H-fluoren-2-yl]-propionamide |
NA |
15488166189 |
NA |
NA |
NA |
NA |
BindingDB |
| TERT |
3-(4-Methyl-piperazin-1-yl)-N-{7-[3-(4-methyl-piperazin-1-yl)-propionylamino]-9-oxo-9H-fluoren-2-yl}-propionamide |
NA |
43651583224 |
NA |
NA |
NA |
NA |
BindingDB |
| TERT |
3-(4-Hydroxy-piperidin-1-yl)-N-{7-[3-(4-hydroxy-piperidin-1-yl)-propionylamino]-9-oxo-9H-fluoren-2-yl}-propionamide |
NA |
18620871367 |
NA |
NA |
NA |
NA |
BindingDB |
| TERT |
3-(2-Ethyl-piperidin-1-yl)-N-{7-[3-(2-ethyl-piperidin-1-yl)-propionylamino]-9-oxo-9H-fluoren-2-yl}-propionamide |
NA |
14125375446 |
NA |
NA |
NA |
NA |
BindingDB |
| TERT |
3-(4-Ethyl-piperazin-1-yl)-N-{7-[3-(4-ethyl-piperazin-1-yl)-propionylamino]-9-oxo-9H-fluoren-2-yl}-propionamide |
NA |
16982436525 |
NA |
NA |
NA |
NA |
BindingDB |
| TERT |
3-(2-Hydroxymethyl-piperidin-1-yl)-N-{7-[3-(2-hydroxymethyl-piperidin-1-yl)-propionylamino]-9-oxo-9H-fluoren-2-yl}-propionamide |
NA |
7943282347 |
NA |
NA |
NA |
NA |
BindingDB |
| TERT |
3-Dimethylamino-N-[7-(3-dimethylamino-propionylamino)-9-oxo-9H-fluoren-2-yl]-propionamide |
NA |
16218100974 |
NA |
NA |
NA |
NA |
BindingDB |
| TERT |
N-[9,10-Dioxo-6-(3-pyrrolidin-1-yl-propionylamino)-9,10-dihydro-anthracen-2-yl]-3-pyrrolidin-1-yl-propionamide |
NA |
1778279410 |
NA |
NA |
NA |
NA |
BindingDB |
| TERT |
3-(2-Methyl-piperidin-1-yl)-N-{7-[3-(2-methyl-piperidin-1-yl)-propionylamino]-9-oxo-9H-fluoren-2-yl}-propionamide |
NA |
12022644346 |
NA |
NA |
NA |
NA |
BindingDB |
| TERT |
{2-[2-(2-Dimethylamino-ethyl)-indolo[3,2-b]quinolin-10-yl]-ethyl}-dimethyl-amine |
NA |
15848931925 |
NA |
NA |
NA |
NA |
BindingDB |
| TERT |
N-(17-methoxy-4,12-diazapentacyclo[11.8.0.02,11.05,10.014,19]henicosa-1(13),2(11),3,5,7,9,14(19),15,17,20-decaen-3-yl)-N',N'-dimethylpropane-1,3-diamine |
NA |
1000000000 |
NA |
NA |
NA |
NA |
BindingDB |
| TERT |
N-(quinolino[3,2-a]acridin-6-ylmethyl)propan-1-amine |
NA |
1445439771 |
NA |
NA |
NA |
NA |
BindingDB |
| TERT |
N',N'-dimethyl-N-(quinolino[3,2-a]acridin-6-ylmethyl)propane-1,3-diamine |
NA |
758577575 |
NA |
NA |
NA |
NA |
BindingDB |
| TERT |
4-[[(3-Amino-5-ethyl-6-phenylphenanthridin-5-ium-8-yl)amino]diazenyl]benzenecarboximidamide |
NA |
18197009|18197008.59 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| TERT |
Camptothecin |
NA |
300000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| TERT |
N-(16-methoxy-4,12-diazapentacyclo[11.8.0.02,11.05,10.014,19]henicosa-1(13),2(11),3,5,7,9,14(19),15,17,20-decaen-3-yl)-N',N'-dimethylethane-1,2-diamine |
NA |
1258925412 |
NA |
NA |
NA |
NA |
BindingDB |
| TERT |
12-[[2-(21-Methyl-10,14-diazapentacyclo[12.7.0.02,10.04,9.015,20]henicosa-1(21),2,4,6,8,15,17,19-octaen-3-yl)acetyl]amino]dodecanoic acid |
NA |
81283051616 |
NA |
NA |
NA |
NA |
BindingDB |
| TERT |
12-[[2-[1-[2-(5-Chloroindol-1-yl)ethyl]indol-3-yl]acetyl]amino]dodecyl cyclohexyl hydrogen phosphate |
NA |
101000 |
NA |
NA |
NA |
NA |
BindingDB |
| TERT |
12-(2-{1-[2-(Naphthalen-1-yloxy)-ethyl]-1H-indol-3-yl}-acetylamino)-dodecanoic acid |
NA |
34673685045 |
NA |
NA |
NA |
NA |
BindingDB |
| TERT |
12-{2-[1-(3-Phenoxy-propyl)-1H-indol-3-yl]-acetylamino}-dodecanoic acid |
NA |
32359365693 |
NA |
NA |
NA |
NA |
BindingDB |