| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| TERT |
12-{2-[1-(3-Cyclohexyloxy-propyl)-1H-indol-3-yl]-acetylamino}-dodecanoic acid |
NA |
67608297539 |
NA |
NA |
NA |
NA |
BindingDB |
| TERT |
12-(2-{1-[3-(3-Methyl-indol-1-yl)-propyl]-1H-indol-3-yl}-acetylamino)-dodecanoic acid |
NA |
19952623150 |
NA |
NA |
NA |
NA |
BindingDB |
| TERT |
12-{2-[1-(3-Indol-1-yl-propyl)-1H-indol-3-yl]-acetylamino}-dodecanoic acid |
NA |
91201083936 |
NA |
NA |
NA |
NA |
BindingDB |
| TERT |
12-{2-[1-(2-Indol-1-yl-ethyl)-1H-indol-3-yl]-acetylamino}-dodecanoic acid |
NA |
40738027780 |
NA |
NA |
NA |
NA |
BindingDB |
| TERT |
12-[[2-(10,13-Diazapentacyclo[11.7.0.02,10.04,9.014,19]icosa-1(20),2,4,6,8,14,16,18-octaen-3-yl)acetyl]amino]dodecanoic acid |
NA |
61659500186 |
NA |
NA |
NA |
NA |
BindingDB |
| TERT |
2-(2,6-Dichloro-benzylsulfanyl)-6-formyl-nicotinonitrile |
NA |
113280 |
NA |
NA |
NA |
NA |
BindingDB |
| TERT |
Topostatin |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| TERT |
3-Pyrrolidin-1-YL-N-[6-(3-pyrrolidin-1-YL-propionylamino)-acridin-3-YL]-propionamide |
NA |
5248074602 |
NA |
NA |
NA |
NA |
BindingDB |
| TERT |
3-N-(2-amino-1,6-dimethylpyrimidin-1-ium-4-yl)-5-methyl-6-(4-methylphenyl)phenanthridin-5-ium-3,8-diamine |
NA |
46773514|46773514.13 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| TERT |
3,11-Difluoro-6,8,13-trimethyl-8H-quino[4,3,2-KL]acridin-13-ium |
NA |
331131121|331131121.5 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| TERT |
Collinomycin |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| TERT |
N,N'-(9,10-Dihydro-9,10-dioxo-2,6-anthracenediyl)bis-1-piperidinepropanamide |
NA |
4466835922 |
NA |
NA |
NA |
NA |
BindingDB |
| TERT |
3,6-Bis(3-piperidinopropionamido)acridine |
NA |
2818382931 |
NA |
NA |
NA |
NA |
BindingDB |
| TERT |
3-(2-Diethylamino-ethoxy)-5a,11a-dihydro-benzo[b]naphtho[2,3-d]furan-6,11-dione |
NA |
6918309709 |
NA |
NA |
NA |
NA |
BindingDB |
| TERT |
3-(azepan-1-yl)-N-[6-[3-(azepan-1-yl)propanoylamino]-9,10-dioxoanthracen-2-yl]propanamide |
NA |
12882495517 |
NA |
NA |
NA |
NA |
BindingDB |
| TERT |
Isometamidium |
NA |
19054607 |
NA |
NA |
NA |
NA |
BindingDB |
| TERT |
[4-[[4-Amino-6-[4-(trimethylazaniumyl)anilino]-1,3,5-triazin-2-yl]amino]phenyl]-trimethylazanium |
NA |
6918309709 |
NA |
NA |
NA |
NA |
BindingDB |
| TERT |
4,8-Dimethyl-3,7,11,15,19,23,27-heptaoxa-31-thia-33,34,35,36,37,38,39,40-octazanonacyclo[28.2.1.12,5.16,9.110,13.114,17.118,21.122,25.126,29]tetraconta-1,4,6(39),8,10(38),12,14(37),16,18(36),20,22(35),24,26(34),28,30(33)-pentadecaene |
NA |
5011872 |
NA |
NA |
NA |
NA |
BindingDB |
| TERT |
6-Hydroxy-3-[1-(4-hydroxy-phenyl)-meth-(E)-ylidene]-3H-benzofuran-2-one |
NA |
400000 |
NA |
NA |
NA |
NA |
TTD |
| TERT |
6-N-[4-[[4-(dimethylamino)-2-methylquinolin-6-yl]amino]-6-methylsulfanyl-1,3,5-triazin-2-yl]-4-N,4-N,2-trimethylquinoline-4,6-diamine |
NA |
40738028 |
NA |
NA |
NA |
NA |
BindingDB |