| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| TDP2 |
4-Benzal-1-methyl-2-phenyl-pyrazol[1,5-a]indol-1-ium;triflate |
NA |
128248 |
NA |
NA |
NA |
NA |
BindingDB |
| TDP2 |
1-Methyl-2-phenyl-4-(3,4,5-trimethoxybenzylidene)pyrazol[1,5-a]indol-1-ium;triflate |
NA |
128332 |
NA |
NA |
NA |
NA |
BindingDB |
| TDP2 |
4-[4-(Dimethylamino)benzylidene]-1-methyl-pyrazol[1,5-a]indol-1-ium-2-carboxylic acid ethyl ester;triflate |
NA |
128246 |
NA |
NA |
NA |
NA |
BindingDB |
| TDP2 |
N,N-diallyl-N'-2,1,3-benzothiadiazol-5-ylthiourea |
NA |
128307 |
NA |
NA |
NA |
NA |
BindingDB |
| TDP2 |
N-[4-[[3-[4-(4-fluorophenyl)piperazin-1-yl]-1,4-dioxonaphthalen-2-yl]sulfamoyl]phenyl]acetamide |
NA |
128309 |
NA |
NA |
NA |
NA |
BindingDB |
| TDP2 |
(S)-Scoulerine |
NA |
128332 |
NA |
NA |
NA |
NA |
BindingDB |
| TDP2 |
N-[3-(1,3-benzodioxol-5-yl)-5-keto-3-pyrazolin-4-yl]-piperonylamide |
NA |
128537 |
NA |
NA |
NA |
NA |
BindingDB |
| TDP2 |
N-[3-(4-methoxyphenyl)-5-oxo-1,2-dihydropyrazol-4-yl]-4-methylbenzamide |
NA |
128332 |
NA |
NA |
NA |
NA |
BindingDB |
| TDP2 |
N-[3-(4-chlorophenyl)-5-keto-3-pyrazolin-4-yl]-4-methyl-benzamide |
NA |
128345 |
NA |
NA |
NA |
NA |
BindingDB |
| TDP2 |
6-hydroxy-2-[4-(2-hydroxyethyl)-3-methyl-5-oxo-2,5-dihydro-1H-pyrazol-1-yl]-5-octyl-4(3H)-pyrimidinone |
NA |
128320 |
NA |
NA |
NA |
NA |
BindingDB |
| TDP2 |
2-({4-[3-(4-Hydroxyphenyl)acryloyl]phenyl}amino)-3-(1-piperidinyl)naphthoquinone |
NA |
128329 |
NA |
NA |
NA |
NA |
BindingDB |
| TDP2 |
Pyrazolo[4,3-c]pyridine-4,6(5H,7H)-dione, 3-amino-2-phenyl- |
NA |
111000 |
NA |
NA |
NA |
NA |
TTD |
| TDP2 |
6-(furan-2-yl)-2-hydroxy-4H-isoquinoline-1,3-dione |
NA |
111000 |
NA |
NA |
NA |
NA |
TTD |
| TDP2 |
|
NA |
128332 |
NA |
NA |
NA |
NA |
BindingDB |
| TDP2 |
7-(Furan-2-Yl)-2-Hydroxyisoquinoline-1,3(2h,4h)-Dione |
NA |
111000 |
NA |
NA |
NA |
NA |
TTD |
| TDP2 |
|
NA |
128289 |
NA |
NA |
NA |
NA |
BindingDB |
| TDP2 |
1-Methyl-4-(4-nitrobenzylidene)-2-phenyl-pyrazol[1,5-a]indol-1-ium;triflate |
NA |
128319 |
NA |
NA |
NA |
NA |
BindingDB |
| TDP2 |
3-amino-2-(4-fluorophenyl)-7H-pyrazolo[4,3-c]pyridine-4,6-dione |
NA |
111000 |
NA |
NA |
NA |
NA |
TTD |
| TDP2 |
N-(4,6-dioxo-2-phenyl-7H-pyrazolo[4,3-c]pyridin-3-yl)acetamide |
NA |
111000 |
NA |
NA |
NA |
NA |
TTD |
| TDP2 |
(4Z)-4-[(5-bromo-2-thiophenyl)methylidene]-5-methyl-2-phenyl-3-pyrazolone |
NA |
128345 |
NA |
NA |
NA |
NA |
BindingDB |