| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| TGM2 |
Dihydroisoxazole, 1c |
430000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| TGM2 |
Dihydroisoxazole, 1d |
390000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| TGM2 |
Sulforaphane |
366000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
| TGM2 |
Dihydroisoxazole, 1i |
910000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| TGM2 |
(E)-3-(4-hydroxyphenyl)-1-pyridin-3-ylprop-2-en-1-one |
NA |
2000000 |
NA |
NA |
NA |
NA |
TTD |
| TGM2 |
(E)-3-(3-hydroxyphenyl)-1-pyridin-3-ylprop-2-en-1-one |
NA |
266000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| TGM2 |
(E)-3-(4-hydroxy-3-methoxyphenyl)-1-pyridin-3-ylprop-2-en-1-one |
NA |
688000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| TGM2 |
Dihydroisoxazole, 1h |
310000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| TGM2 |
Dihydroisoxazole, 1g |
240000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| TGM2 |
Dihydroisoxazole, 2a |
1300000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| TGM2 |
Dihydroisoxazole, 2b |
260000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| TGM2 |
Dihydroisoxazole, 3a |
2700000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| TGM2 |
Isatin |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| TGM2 |
(2S)-6-(1,3-diethyl-4,5-dimethylimidazol-1-ium-2-yl)sulfanyl-5-oxo-2-[[(2S)-3-phenyl-2-(phenylmethoxycarbonylamino)propanoyl]amino]hexanoic acid;bromide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| TGM2 |
(2S)-6-(1,3-diethyl-4,5-dimethylimidazol-1-ium-2-yl)sulfanyl-5-oxo-2-[[2-(phenylmethoxycarbonylamino)acetyl]amino]hexanoic acid;bromide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| TGM2 |
(2S)-5-oxo-2-[[(2S)-3-phenyl-2-(phenylmethoxycarbonylamino)propanoyl]amino]-6-(1,4,5-trimethyl-3-propylimidazol-1-ium-2-yl)sulfanylhexanoic acid;bromide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| TGM2 |
(2S)-5-oxo-2-[[2-(phenylmethoxycarbonylamino)acetyl]amino]-6-(1,4,5-trimethyl-3-propylimidazol-1-ium-2-yl)sulfanylhexanoic acid;bromide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| TGM2 |
(2S)-5-oxo-2-[[(2S)-3-phenyl-2-(phenylmethoxycarbonylamino)propanoyl]amino]-6-(1,4,5-trimethyl-3-phenylimidazol-1-ium-2-yl)sulfanylhexanoic acid;bromide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| TGM2 |
(2S)-5-oxo-2-[[2-(phenylmethoxycarbonylamino)acetyl]amino]-6-(1,4,5-trimethyl-3-phenylimidazol-1-ium-2-yl)sulfanylhexanoic acid;bromide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| TGM2 |
(2S)-6-(1-benzyl-3,4,5-trimethylimidazol-3-ium-2-yl)sulfanyl-5-oxo-2-[[(2S)-3-phenyl-2-(phenylmethoxycarbonylamino)propanoyl]amino]hexanoic acid;bromide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |