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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
TGM2 (2S)-6-(1-benzyl-3,4,5-trimethylimidazol-3-ium-2-yl)sulfanyl-5-oxo-2-[[2-(phenylmethoxycarbonylamino)acetyl]amino]hexanoic acid;bromide NA 200000 NA NA NA NA TTD
TGM2 (E)-3-(3-ethoxy-4-hydroxyphenyl)-1-pyridin-3-ylprop-2-en-1-one NA 484000 NA NA NA NA BindingDB|TTD
THRA 2-(3,5-Dibromo-4-ethoxyphenyl)acetic acid NA 160000 NA NA NA NA BindingDB|TTD
THRB Limonene, (+/-)- NA NA NA NA 794328 NA PubChem
THRB Bithionol NA NA NA NA 125892 NA PubChem
THRB Chlormezanone NA NA NA NA 112202 NA PubChem
THRB Tacrine Hydrochloride NA NA NA NA 1000000 NA PubChem
THRB Silybin NA NA NA NA 125892 NA PubChem
THRB Emodin NA NA NA NA 112202 NA PubChem
THRB Indigotindisulfonic acid NA NA NA NA 354813 NA PubChem
THRB Mesalamine NA NA NA NA 125892 NA PubChem
THRB Resveratrol NA NA NA NA 112202 NA PubChem
THRB Levothyroxine NA NA NA NA 112202 NA PubChem
THRB Chlorobutanol NA NA NA NA 112202 NA PubChem
THRB Atorvastatin NA NA NA NA 112202 NA PubChem
THRB Cytarabine NA NA NA NA 2238720 NA PubChem
THRB Diltiazem Hydrochloride NA NA NA NA 2511890 NA PubChem
THRB 2-Phenylphenol NA NA NA NA 281838|251189 NA PubChem
THRB 1H-Imidazole, 1-[1-[[4-chloro-2-(trifluoromethyl)phenyl]imino]-2-propoxyethyl]- NA NA NA NA 125892 NA PubChem
THRB Nandrolone NA NA NA NA 125892 NA PubChem