GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
TMPRSS6 |
Tert-butyl 4-[[2-[(3-carbamimidoylphenyl)sulfonylamino]acetyl]amino]benzoate;2,2,2-trifluoroacetic acid |
137000 |
NA |
NA |
NA |
NA |
NA |
TTD |
TMPRSS6 |
Tert-butyl 3-[4-[(3-carbamimidoylphenyl)sulfonylamino]butanoylamino]benzoate;2,2,2-trifluoroacetic acid |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
TMPRSS6 |
4-[[2-[(4-Carbamimidoylphenyl)sulfonylamino]acetyl]amino]benzoic acid;2,2,2-trifluoroacetic acid |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
TMPRSS6 |
3-[[2-[(4-Carbamimidoylphenyl)sulfonylamino]acetyl]amino]benzoic acid;2,2,2-trifluoroacetic acid |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
TMPRSS6 |
4-[3-[(4-Carbamimidoylphenyl)sulfonylamino]propanoylamino]benzoic acid;2,2,2-trifluoroacetic acid |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
TMPRSS6 |
3-[3-[(4-Carbamimidoylphenyl)sulfonylamino]propanoylamino]benzoic acid;2,2,2-trifluoroacetic acid |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
TMPRSS6 |
4-[4-[(4-Carbamimidoylphenyl)sulfonylamino]butanoylamino]benzoic acid;2,2,2-trifluoroacetic acid |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
TMPRSS6 |
3-[4-[(4-Carbamimidoylphenyl)sulfonylamino]butanoylamino]benzoic acid;2,2,2-trifluoroacetic acid |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
TMPRSS6 |
4-[[2-[(3-Carbamimidoylphenyl)sulfonylamino]acetyl]amino]benzoic acid;2,2,2-trifluoroacetic acid |
139000 |
NA |
NA |
NA |
NA |
NA |
TTD |
TMPRSS6 |
3-[[2-[(3-Carbamimidoylphenyl)sulfonylamino]acetyl]amino]benzoic acid;2,2,2-trifluoroacetic acid |
207000 |
NA |
NA |
NA |
NA |
NA |
TTD |
TMPRSS6 |
3-[3-[(3-Carbamimidoylphenyl)sulfonylamino]propanoylamino]benzoic acid;2,2,2-trifluoroacetic acid |
208000 |
NA |
NA |
NA |
NA |
NA |
TTD |
TMPRSS6 |
4-[4-[(3-Carbamimidoylphenyl)sulfonylamino]butanoylamino]benzoic acid;2,2,2-trifluoroacetic acid |
217000 |
NA |
NA |
NA |
NA |
NA |
TTD |
TMPRSS6 |
3-[4-[(3-Carbamimidoylphenyl)sulfonylamino]butanoylamino]benzoic acid;2,2,2-trifluoroacetic acid |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
TMPRSS6 |
[Amino-[3-[[4-(4-carboxyanilino)-4-oxobutyl]sulfamoyl]phenyl]methylidene]azanium |
217000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
TMPRSS6 |
[Amino-[3-[[3-(3-carboxyanilino)-3-oxopropyl]sulfamoyl]phenyl]methylidene]azanium |
208000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
TMPRSS6 |
[Amino-[3-[[2-(3-carboxyanilino)-2-oxoethyl]sulfamoyl]phenyl]methylidene]azanium |
207000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
TMPRSS6 |
[Amino-[3-[[2-(4-carboxyanilino)-2-oxoethyl]sulfamoyl]phenyl]methylidene]azanium |
139000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
TMPRSS6 |
[Amino-[3-[[2-[4-[(2-methylpropan-2-yl)oxycarbonyl]anilino]-2-oxoethyl]sulfamoyl]phenyl]methylidene]azanium |
137000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
TMPRSS6 |
[Amino-[3-[[2-(naphthalen-1-ylsulfonylamino)acetyl]amino]phenyl]methylidene]azanium |
163000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
TMPRSS6 |
[Amino-[3-[[2-(naphthalen-2-ylsulfonylamino)acetyl]amino]phenyl]methylidene]azanium |
163000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |